| 货号 (SKU) | 包装规格 | 是否现货 | 价格 | 数量 |
|---|---|---|---|---|
| R105077-250mg |
250mg |
现货  |
|
| 英文别名 | C23H22O6 | EINECS 201-501-9 | Spectrum4_001638 | Derris resins | Liquid Derris | (1S,6R,13S)-16,17-dimethoxy-6-prop-1-en-2-yl-2,7,20-trioxapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),9,14,16,18-hexaen-12-one | (2R,6aS,12aS)-8,9-Dimethoxy-2-(pr |
|---|---|
| 规格或纯度 | 分析标准品, ≥96% |
| 英文名称 | Rotenone |
| 生化机理 | 鱼藤酮是烟酰胺腺嘌呤二核苷酸（NADH）：泛醌氧化还原酶线上粒体电子传递的一种抑制剂。它能够很容易的通过节肢动物的外骨骼被吸收，但皮肤或哺乳动物的胃肠道的吸收则不佳。鱼藤酮作为一种神经毒素能产生帕金森样症状，从而作为一种动物模型用于作为病因和干预措施的研究。 |
| 应用 | 线粒体电子传递的抑制剂 |
| 储存温度 | 避光,充氩 |
| 运输条件 | 常规运输 |
| 产品介绍 |
难溶于水,易溶于极性有机溶剂,在氯仿中溶解度最大(472g/L) ,遇碱消旋。易氧化尤其在光或碱存在下氧化快而失去杀虫活性,在干燥情况下比较稳定。对光和空气敏感， 线粒体电子传递的抑制剂。 应用： 鱼藤酮已用于： |
| 纯度 | ≥96% |
| 作用机制 | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | 参考文献 |
|---|
| EC号 | 201-501-9 |
|---|---|
| 分子类型 | 小分子 |
| IIUPAC Name | (1S,6R,13S)-16,17-dimethoxy-6-prop-1-en-2-yl-2,7,20-trioxapentacyclo[11.8.0.03,11.04,8.014,19]henicosa-3(11),4(8),9,14,16,18-hexaen-12-one |
| INCHI | 1S/C23H22O6/c1-11(2)16-8-14-15(28-16)6-5-12-22(24)21-13-7-18(25-3)19(26-4)9-17(13)27-10-20(21)29-23(12)14/h5-7,9,16,20-21H,1,8,10H2,2-4H3/t16-,20-,21+/m1/s1 |
| InChi Key | JUVIOZPCNVVQFO-HBGVWJBISA-N |
| Smiles | CC(=C)C1CC2=C(O1)C=CC3=C2OC4COC5=CC(=C(C=C5C4C3=O)OC)OC |
| Isomeric SMILES | CC(=C)[C@H]1CC2=C(O1)C=CC3=C2O[C@@H]4COC5=CC(=C(C=C5[C@@H]4C3=O)OC)OC |
| PubChem CID | 6758 |
| UN Number | 2588 |
| Packing Group | I |
| 分子量 | 394.42 |
| Beilstein号 | 6773081 |
| 密度 | 1.27 |
|---|---|
| 敏感性 | 对光和空气敏感 |
| 沸点 | 210-220°C |
| 熔点 | 159-164°C |
| 分子量 | 394.400 g/mol |
| XLogP3 | 4.100 |
| 氢键供体数Hydrogen Bond Donor Count | 0 |
| 氢键受体数Hydrogen Bond Acceptor Count | 6 |
| 可旋转键计数Rotatable Bond Count | 3 |
| 精确质量Exact Mass | 394.142 Da |
| 单同位素质量Monoisotopic Mass | 394.142 Da |
| 拓扑极表面积Topological Polar Surface Area | 63.200 Ų |
| 重原子数Heavy Atom Count | 29 |
| 形式电荷Formal Charge | 0 |
| 复杂度Complexity | 664.000 |
| 同位素原子数Isotope Atom Count | 0 |
| 定义的原子立体中心计数Defined Atom Stereocenter Count | 3 |
| 未定义的原子立体中心计数Undefined Atom Stereocenter Count | 0 |
| 定义的键立体中心计数Defined Bond Stereocenter Count | 0 |
| 未定义的键立体中心计数Undefined Bond Stereocenter Count | 0 |
| 所有立体化学键的总数The total count of all stereochemical bonds | 0 |
| 共价键合单元计数Covalently-Bonded Unit Count | 1 |
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