还原型 S-己基-L-谷胱甘肽

谷胱甘肽S-转移酶抑制剂

6篇引用文献

COA

级别和纯度:

≥98%

CAS编号: 24425-56-7
分子式: C₁₆H₂₉N₃O₆S
分子量: 391.48
Beilstein号: 5629635
MDL号: MFCD00056735
PubChem编号: 97536
PubChem SID: 504756373

有货

库存信息

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库存信息

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货号 (SKU)	包装规格	是否现货	价格	数量
H121370-25mg	25mg	现货
H121370-100mg	100mg	现货

查看相关系列

Amino Acid/Protein Metabolism (4559) 多肽 (100)

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基本描述

别名	还原型 S-己基-L-谷胱甘肽 \| S -己基谷胱甘肽
英文别名	BDBM50095998 \| 1ydk \| C02886 \| GTPL1941 \| S-Hexyl-L-glutathione (H-L-gGlu-Cys(hexyl)-Gly-OH) \| MFCD00056735 \| NSC-131114 \| (2S)-2-azanyl-5-[[(2R)-3-hexylsulfanyl-1-(2-hydroxy-2-oxoethylamino)-1-oxidanylidene-propan-2-yl]amino]-5-oxidanylidene-pentanoic ac
规格或纯度	≥98%
英文名称	S-Hexylglutathione
生化机理	S-己基谷胱甘肽可用作谷胱甘肽-S-转移酶和谷胱甘肽过氧化物酶的亲和层析配体。S-己基谷胱甘肽还可用作抑制剂，用于研究线粒体膜结合谷胱甘肽转移酶（mtMGST1）等酶的特异性和动力学。与 G 位点结合，稳定 GST 免受尿素的影响。与巨噬细胞迁移抑制因子结合（K d = 2.5 mM）。
应用	Ligand useful for affinity chromatography of glutathione-S-transferase and glutathione peroxidase.
储存温度	2-8°C储存
运输条件	冰袋运输
备注	如果有可能，您尽量在使用的当天配置溶液，并在当天使用完它。但是，如果您需要预先配制储备溶液，我们建议您将溶液等份保存在-20°C的密封小瓶中。通常，它们最多可以使用一个月。在使用前和打开样品瓶之前，我们建议您让您的产品在室温下平衡至少1小时。需要更多关于溶解度，用法和处理的建议吗？请访问我们的常见问题（FAQ）页面以获取更多详细信息。
产品介绍	用于谷胱甘肽-S-转移酶和谷胱甘肽过氧化物酶的亲和色谱法的配体。
纯度	≥98%

关联靶点（人）

GSTA1 Tchem 谷胱甘肽S-转移酶A1(Glutathione S-transferase A1) (0 活性数据)

点击查看靶蛋白信息： GSTA1

活性类型	活性值-log(M)	作用机制	期刊	参考文献(PubMed IDs)

作用机制

作用机制	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	参考文献

名称和识别符

PubChem SID	504756373
分子类型	小分子
IIUPAC Name	(2S)-2-amino-5-[[(2R)-1-(carboxymethylamino)-3-hexylsulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid
INCHI	1S/C16H29N3O6S/c1-2-3-4-5-8-26-10-12(15(23)18-9-14(21)22)19-13(20)7-6-11(17)16(24)25/h11-12H,2-10,17H2,1H3,(H,18,23)(H,19,20)(H,21,22)(H,24,25)/t11-,12-/m0/s1
InChi Key	HXJDWCWJDCOHDG-RYUDHWBXSA-N
Smiles	CCCCCCSCC(C(=O)NCC(=O)O)NC(=O)CCC(C(=O)O)N
Isomeric SMILES	CCCCCCSC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N
分子量	391.48
Beilstein号	5629635
Reaxy-Rn	24735187
Reaxys-RN link address	https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=24735187&ln=

化学和物理性质

熔点	200-202 °C
分子量	391.500 g/mol
XLogP3	-1.800
氢键供体数Hydrogen Bond Donor Count	5
氢键受体数Hydrogen Bond Acceptor Count	8
可旋转键计数Rotatable Bond Count	15
精确质量Exact Mass	391.178 Da
单同位素质量Monoisotopic Mass	391.178 Da
拓扑极表面积Topological Polar Surface Area	184.000 Å²
重原子数Heavy Atom Count	26
形式电荷Formal Charge	0
复杂度Complexity	475.000
同位素原子数Isotope Atom Count	0
定义的原子立体中心计数Defined Atom Stereocenter Count	2
未定义的原子立体中心计数Undefined Atom Stereocenter Count	0
定义的键立体中心计数Defined Bond Stereocenter Count	0
未定义的键立体中心计数Undefined Bond Stereocenter Count	0
所有立体化学键的总数The total count of all stereochemical bonds	0
共价键合单元计数Covalently-Bonded Unit Count	1

安全和危险性（GHS）

WGK Germany	3

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找到10个结果

批号(Lot Number)	证书类型	货号
I2511676	分析证书	H121370
I2511679	分析证书	H121370
K2422582	分析证书	H121370
K2422587	分析证书	H121370
H2423342	分析证书	H121370
H2423335	分析证书	H121370
H2423343	分析证书	H121370
J1923170	分析证书	H121370
C2212337	分析证书	H121370
C2212342	分析证书	H121370

此产品的引用文献

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引用文献

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