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SHU9119,TFA - ≥95%, high purity , CAS No.168482-23-3(free base), Agonist of MC 1 receptor;Antagonist of MC 3 receptor;Antagonist of MC 4 receptor;Agonist of MC 5 receptor

In stock
Item Number
S275436
Grouped product items
SKU Size
Availability
Price Qty
S275436-1mg
1mg
3
$84.90
S275436-5mg
5mg
3
$338.90
S275436-10mg
10mg
3
$541.90
S275436-25mg
25mg
3
$948.90
S275436-50mg
50mg
2
$1,517.90

Potent melanocortin 3 and 4 (MC 3 and MC 4 ) receptor antagonist

Basic Description

Synonyms SHU 9119
Specifications & Purity Moligand™, ≥95%
Biochemical and Physiological Mechanisms Potent melanocortin 3 and 4 (MC 3 and MC 4 ) receptor antagonist (IC 50 values are 0.23 and 0.06 nM, respectively). Also shows MC 5 partial agonist activity (EC 50 = 0.12 nM). Dose-dependently increases food intake following central administration.
Storage Temp Store at -20°C,Desiccated
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Grade Moligand™
Action Type AGONIST, ANTAGONIST
Mechanism of action Agonist of MC 1 receptor;Antagonist of MC 3 receptor;Antagonist of MC 4 receptor;Agonist of MC 5 receptor

Associated Targets(Human)

MC5R Tchem Melanocortin receptor 5 (0 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
MC4R Tclin Melanocortin receptor 4 (0 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
MC3R Tchem Melanocortin receptor 3 (0 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
MC1R Tclin Melanocyte-stimulating hormone receptor (0 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)

Names and Identifiers

Molecular Weight 1074.25(free base)

Certificates(CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Find and download the COA for your product by matching the lot number on the packaging.

10 results found

Lot Number Certificate Type Date Item
C2425491 Certificate of Analysis Jun 17, 2025 S275436
C2425502 Certificate of Analysis Jun 17, 2025 S275436
C2425503 Certificate of Analysis Jun 17, 2025 S275436
C2425504 Certificate of Analysis Jun 17, 2025 S275436
C2425492 Certificate of Analysis Jun 17, 2025 S275436
C2425472 Certificate of Analysis Jan 15, 2025 S275436
C2425471 Certificate of Analysis Jan 15, 2025 S275436
C2425473 Certificate of Analysis Jan 15, 2025 S275436
C2425474 Certificate of Analysis Jan 15, 2025 S275436
C2425475 Certificate of Analysis Jan 15, 2025 S275436

Chemical and Physical Properties

Solubility Soluble in water

Solution Calculators

Reviews

Customer Reviews

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