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(R)-PS210 - 98%, high purity , CAS No.1410101-89-1

    Grade & Purity:
  • ≥98%
In stock
Item Number
P650497
Grouped product items
SKU Size
Availability
Price Qty
P650497-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$250.90
P650497-10mg
10mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$390.90
P650497-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$780.90
P650497-50mg
50mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,250.90
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Basic Description

Specifications & Purity ≥98%
Biochemical and Physiological Mechanisms (R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC 50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket ofxa0PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-inter
Storage Temp Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Product Description

(R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC 50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket of PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment

In Vitro

(R)-PS210 displays an AC 50 value of 1.8 μM towards PDK1 in a Cell-Free Kinase Activity Assay. And the maximum activation of PDK1 compared to DMSO control of (R)-PS210 is 5.5 fold. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:AC50: 1.8 μM (PDK1)

Names and Identifiers

Smiles O=C(O)C([C@H](C1=CC=CC=C1)CC(C2=CC=C(C(F)(F)F)C=C2)=O)C(O)=O
Molecular Weight 380.31

Certificates(CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Chemical and Physical Properties

Solubility DMSO : 230 mg/mL (604.77 mM; Need ultrasonic)

Solution Calculators

Reviews

Customer Reviews

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