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| SKU | Size | Availability |
Price | Qty |
|---|---|---|---|---|
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P650708-5mg
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5mg |
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
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$50.90
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P650708-10mg
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10mg |
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
|
$70.90
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P650708-50mg
|
50mg |
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
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$280.90
|
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P650708-100mg
|
100mg |
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
|
$480.90
|
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| Synonyms | 2-Phenyl-4-(2-(piperidin-4-yl)ethyl)quinoline | PK-8165 |
|---|---|
| Specifications & Purity | Moligand™, ≥99% |
| Biochemical and Physiological Mechanisms | Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. |
| Storage Temp | Store at -20°C |
| Shipped In |
Ice chest + Ice pads This product requires cold chain shipping. Ground and other economy services are not available. |
| Grade | Moligand™ |
| Product Description |
Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity In Vivo Intravenously administered pipequaline exerts a partial suppression of activations by kainate, glutamate and acetylcholine. Microiontophoretic applications of pipequaline reduces the neuronal activation by kainate. Pipequaline produces dose-related decreases in motor activity. Pipequaline produces significant dose-related decreases in the number of head-dips made. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Form:Solid IC50& Target:Benzodiazepine receptor |
| Mechanism of Action | Action Type | target ID | Target Name | Target Type | Target Organism | Binding Site Name | References |
|---|
| Smiles | C1CNCCC1CCC2=CC(=NC3=CC=CC=C32)C4=CC=CC=C4 |
|---|---|
| Isomeric SMILES | C1CNCCC1CCC2=CC(=NC3=CC=CC=C32)C4=CC=CC=C4 |
| PubChem CID | 71219 |
| Molecular Weight | 316.44 |
| Solubility | DMSO : ≥ 32 mg/mL (101.13 mM) |
|---|---|
| Molecular Weight | 316.400 g/mol |
| XLogP3 | 5.000 |
| Hydrogen Bond Donor Count | 1 |
| Hydrogen Bond Acceptor Count | 2 |
| Rotatable Bond Count | 4 |
| Exact Mass | 316.194 Da |
| Monoisotopic Mass | 316.194 Da |
| Topological Polar Surface Area | 24.900 Ų |
| Heavy Atom Count | 24 |
| Formal Charge | 0 |
| Complexity | 370.000 |
| Isotope Atom Count | 0 |
| Defined Atom Stereocenter Count | 0 |
| Undefined Atom Stereocenter Count | 0 |
| Defined Bond Stereocenter Count | 0 |
| Undefined Bond Stereocenter Count | 0 |
| The total count of all stereochemical bonds | 0 |
| Covalently-Bonded Unit Count | 1 |
Starting at $55.90
Starting at $1,515.90