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Basic Information
ID: ALA4325019
Type: Binding
Description: Protac activity against VHL/AR in AR-positive human LNCAP cells assessed as reduction in TMPRSS2 mRNA expression level incubated for 24 hrs by qRT-PCR analysis relative to N-((1r,3r)-3-(3-Chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)-1-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
Format: BAO_0000219
Organism: Homo sapiens
Cell type: LNCaP
Target: VHL/Androgen receptor(ALA4523730)
Document: ALA4321866
Protac activity against VHL/AR in AR-positive human LNCAP cells assessed as reduction in TMPRSS2 mRNA expression level incubated for 24 hrs by qRT-PCR analysis relative to N-((1r,3r)-3-(3-Chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)-1-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4325019
FC
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 915.53 | 7.36 | 7.36 |
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