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Phosphoglycerate Dehydrogenase (PHGDH)

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12 Items

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  1. PKUMDL WQ 2101
      Grade & Purity: 
    • ≥98%(HPLC)
    Cas Number: 304481-72-9        Compound CID:  135781546
    Formula:  C14H11N3O6        Molecular Weight: 317.25
    IUPAC Name:  2,4-dihydroxy-N-[(Z)-(2-hydroxy-5-nitrophenyl)methylideneamino]benzamide
    SMILES:  C1=CC(=C(C=C1[N+](=O)[O-])C=NNC(=O)C2=C(C=C(C=C2)O)O)O
    InChIKey: OXONIXZPWKJHMW-CHHVJCJISA-N
    InChI:  InChI=1S/C14H11N3O6/c18-10-2-3-11(13(20)6-10)14(21)16-15-7-8-5-9(17(22)23)1-4-12(8)19/h1-7,18-20H,(H,16,21)/b15-7-
    Synonyms: 2,4-Dihydroxy-N'-(2-hydroxy-5-nitrobenzylidene)benzohydrazide | PKUMDL-WQ-2101
  2. D-3-Phosphoglyceric acid disodium salt
      Grade & Purity: 
    • ≥98%
    Cas Number: 80731-10-8
    Formula:  C3H5O7P・2Na        Molecular Weight: 230.02
    IUPAC Name:  disodium;(2R)-2-hydroxy-3-[hydroxy(oxido)phosphoryl]oxypropanoate
    SMILES:  [Na+].[Na+].O[C@H](COP(O)([O-])=O)C([O-])=O
    InChIKey: RGCJWQYUZHTJBE-YBBRRFGFSA-L
    InChI:  InChI=1S/C3H7O7P.2Na/c4-2(3(5)6)1-10-11(7,8)9;;/h2,4H,1H2,(H,5,6)(H2,7,8,9);;/q;2*+1/p-2/t2-;;/m1../s1
    Synonyms: D-Glycerate 3-phosphate disodium salt | (-)-Disodium D-3-phosphoglycerate | 3-Phospho-D-glyceric acid disodium
  3. D-(-)-3-Phosphoglyceric acid disodium salt
      Grade & Purity: 
    • ≥93%
    Cas Number: 80731-10-8
    Formula:  C3H5O7P・2Na        Molecular Weight: 230.02
    IUPAC Name:  disodium;(2R)-2-hydroxy-3-[hydroxy(oxido)phosphoryl]oxypropanoate
    SMILES:  [Na+].[Na+].O[C@H](COP(O)([O-])=O)C([O-])=O
    InChIKey: RGCJWQYUZHTJBE-YBBRRFGFSA-L
    InChI:  InChI=1S/C3H7O7P.2Na/c4-2(3(5)6)1-10-11(7,8)9;;/h2,4H,1H2,(H,5,6)(H2,7,8,9);;/q;2*+1/p-2/t2-;;/m1../s1
    Synonyms: Sodium (R)-2-carboxy-2-hydroxyethyl phosphate | 4-HEXYLOXY-BENZOICACIDHYDRAZIDE | PROPANOIC ACID,2-HYDROXY-3-(PHOSPHO...
  4. PKUMDL WQ 2201
      Grade & Purity: 
    • ≥98%(HPLC)
    Cas Number: 592474-91-4        Compound CID:  6875399
    Formula:  C15H14ClN3O3S        Molecular Weight: 351.81
    IUPAC Name:  2-chloro-4-[5-[(E)-(ethylcarbamothioylhydrazinylidene)methyl]furan-2-yl]benzoic acid
    SMILES:  CCNC(=S)NN=CC1=CC=C(O1)C2=CC(=C(C=C2)C(=O)O)Cl
    InChIKey: XPACBFAEZIPDRT-QGMBQPNBSA-N
    InChI:  InChI=1S/C15H14ClN3O3S/c1-2-17-15(23)19-18-8-10-4-6-13(22-10)9-3-5-11(14(20)21)12(16)7-9/h3-8H,2H2,1H3,(H,20,21)(H2,17,19,23)/b18-8+
    Synonyms: 2-Chloro-4-[5-[[2-[(ethylamino)thioxomethyl]hydrazinylidene]methyl]-2-furanyl]benzoic acid
  5. CBR 5884
      Grade & Purity: 
    • ≥98%(HPLC)
    Cas Number: 681159-27-3
    Formula:  C14H12N2O4S2        Molecular Weight: 336.39
    IUPAC Name:  ethyl 5-(furan-2-carbonylamino)-3-methyl-4-thiocyanatothiophene-2-carboxylate
    SMILES:  CCOC(=O)C1=C(C(=C(S1)NC(=O)C2=CC=CO2)SC#N)C
    InChIKey: QBVIRPJBDIZKBC-UHFFFAOYSA-N
    InChI:  InChI=1S/C14H12N2O4S2/c1-3-19-14(18)11-8(2)10(21-7-15)13(22-11)16-12(17)9-5-4-6-20-9/h4-6H,3H2,1-2H3,(H,16,17)
    Synonyms: 5-[(2-Furanylcarbonyl)amino]-3-methyl-4-thiocyanato-2-thiophenecarboxylic acid ethyl ester
  6. CBR 5884
      Grade & Purity: 
    • 10mM in DMSO
    Cas Number: 681159-27-3
    Formula:  C14H12N2O4S2        Molecular Weight: 336.39
    IUPAC Name:  ethyl 5-(furan-2-carbonylamino)-3-methyl-4-thiocyanatothiophene-2-carboxylate
    SMILES:  CCOC(=O)C1=C(C(=C(S1)NC(=O)C2=CC=CO2)SC#N)C
    InChIKey: QBVIRPJBDIZKBC-UHFFFAOYSA-N
    InChI:  InChI=1S/C14H12N2O4S2/c1-3-19-14(18)11-8(2)10(21-7-15)13(22-11)16-12(17)9-5-4-6-20-9/h4-6H,3H2,1-2H3,(H,16,17)
    Synonyms: Ethyl 5-[(2-furanylcarbonyl)amino]-3-methyl-4-thiocyanato-2-thiophenecarboxylate
  7. NCT-503
      Grade & Purity: 
    • ≥98%
    Cas Number: 1916571-90-8
    Formula:  C20H23F3N4S        Molecular Weight: 408.48
    IUPAC Name:  N-(4,6-dimethylpyridin-2-yl)-4-[[4-(trifluoromethyl)phenyl]methyl]piperazine-1-carbothioamide
    SMILES:  CC1=CC(=NC(=C1)NC(=S)N2CCN(CC2)CC3=CC=C(C=C3)C(F)(F)F)C
    InChIKey: PJNSZIQUFLWRLH-UHFFFAOYSA-N
    InChI:  InChI=1S/C20H23F3N4S/c1-14-11-15(2)24-18(12-14)25-19(28)27-9-7-26(8-10-27)13-16-3-5-17(6-4-16)20(21,22)23/h3-6,11-12H,7-10,13H2,1-2H3,(H,24,25,28)
    Synonyms: 1-​Piperazinecarbothioa​mide,N-​(4,​6-​dimethyl-​2-​pyridinyl)​-​4-​[[4-​(trifluoromethyl)​phenyl]​methyl]​-
  8. PHGDH-inactive
      Grade & Purity: 
    • ≥99%
    Cas Number: 1914971-16-6        Compound CID:  49853203
    Formula:  C17H21N5S        Molecular Weight: 327.45
    IUPAC Name:  N-(4,6-dimethylpyridin-2-yl)-4-pyridin-4-ylpiperazine-1-carbothioamide
    SMILES:  CC1=CC(=NC(=C1)NC(=S)N2CCN(CC2)C3=CC=NC=C3)C
    InChIKey: ITLPIAAGIQAGRA-UHFFFAOYSA-N
    InChI:  InChI=1S/C17H21N5S/c1-13-11-14(2)19-16(12-13)20-17(23)22-9-7-21(8-10-22)15-3-5-18-6-4-15/h3-6,11-12H,7-10H2,1-2H3,(H,19,20,23)
  9. NCT-502
      Grade & Purity: 
    • ≥99%
    Cas Number: 1542213-00-2        Compound CID:  49853368
    Formula:  C18H20F3N5S        Molecular Weight: 395.45
    IUPAC Name:  N-(4,6-dimethylpyridin-2-yl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazine-1-carbothioamide
    SMILES:  CC1=CC(=NC(=C1)NC(=S)N2CCN(CC2)C3=NC=C(C=C3)C(F)(F)F)C
    InChIKey: HHKPPMSUPATMKP-UHFFFAOYSA-N
    InChI:  InChI=1S/C18H20F3N5S/c1-12-9-13(2)23-15(10-12)24-17(27)26-7-5-25(6-8-26)16-4-3-14(11-22-16)18(19,20)21/h3-4,9-11H,5-8H2,1-2H3,(H,23,24,27)
  10. BI-4916
      Grade & Purity: 
    • ≥98%
    Cas Number: 2244451-48-5        Compound CID:  138911337
    Formula:  C23H24Cl2N2O6S        Molecular Weight: 527.42
    IUPAC Name:  ethyl 2-[4-[(1S)-1-[(4,5-dichloro-1,6-dimethylindole-2-carbonyl)amino]-2-hydroxyethyl]phenyl]sulfonylacetate
    SMILES:  CCOC(=O)CS(=O)(=O)C1=CC=C(C=C1)C(CO)NC(=O)C2=CC3=C(N2C)C=C(C(=C3Cl)Cl)C
    InChIKey: HCDAVCLCBXIYPW-QGZVFWFLSA-N
    InChI:  InChI=1S/C23H24Cl2N2O6S/c1-4-33-20(29)12-34(31,32)15-7-5-14(6-8-15)17(11-28)26-23(30)19-10-16-18(27(19)3)9-13(2)21(24)22(16)25/h5-10,17,28H,4,11-12H2,show more
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