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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4206625 |
12 | Activity | 0 | ALA4183898 | Active | Homo sapiens | |||||
| 2. |
ALA4213959 |
11 | Activity | 0 | ALA4183898 | Not Active | Homo sapiens | |||||
| 3. |
ALA4218881 |
10 | Activity | 0 | ALA4183898 | Active | Homo sapiens | |||||
| 4. |
ALA4216822 |
9 | Activity | 0 | ALA4183898 | Active | Homo sapiens | |||||
| 5. |
ALA4206625 |
12 | Activity | 0 | ALA4183897 | Active | Homo sapiens | |||||
| 6. |
ALA4213959 |
11 | Activity | 0 | ALA4183897 | Active | Homo sapiens | |||||
| 7. |
ALA4218881 |
10 | Activity | 0 | ALA4183897 | Active | Homo sapiens | |||||
| 8. |
ALA4216822 |
9 | Activity | 0 | ALA4183897 | Active | Homo sapiens | |||||
| 9. |
MRS 2578 |
SID26753205 | IC50 | = | 0.037 | uM | ALA4186855 | 7.43 | nM | Homo sapiens | ||
| 10. |
ALA5272895 |
58; MRS2567 | IC50 | = | 100 | nM | ALA5257758 | 7.00 | nM | Homo sapiens | ||
| 11. |
MRS 2578 |
SID26753205 | IC50 | = | 37 | nM | ALA5257758 | 7.43 | nM | Homo sapiens | ||
| 12. |
UDP |
3 | EC50 | = | 0.3 | uM | ALA5257757 | 6.52 | nM | Homo sapiens |