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Chemical synthesis

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  1. Citral, Channel blocker of TRPV2;Activator of TRPV3
      Grade & Purity: 
    • Moligand™
    • ≥97%
    • mixture of cis and trans
    Cas Number: 5392-40-5
    Formula:  C10H16O        Molecular Weight: 152.24
    IUPAC Name:  (2E)-3,7-dimethylocta-2,6-dienal
    SMILES:  CC(=CCCC(=CC=O)C)C
    InChIKey: WTEVQBCEXWBHNA-JXMROGBWSA-N
    InChI:  InChI=1S/C10H16O/c1-9(2)5-4-6-10(3)7-8-11/h5,7-8H,4,6H2,1-3H3/b10-7+
    Synonyms: EINECS 226-394-6 | LMPR0102010003 | alpha -Citral | beta-Geranial | geranal | (2E)-3,7-Dimethyl-2,6-octadienal | UNII...
  2. Flavone, Antagonist of A 1 receptor;Antagonist of A 2A receptor;Antagonist of A 3 receptor
    Cas Number: 525-82-6
    Formula:  C15H10O2        Molecular Weight: 222.24
    IUPAC Name:  2-phenylchromen-4-one
    SMILES:  C1=CC=C(C=C1)C2=CC(=O)C3=CC=CC=C3O2
    InChIKey: VHBFFQKBGNRLFZ-UHFFFAOYSA-N
    InChI:  InChI=1S/C15H10O2/c16-13-10-15(11-6-2-1-3-7-11)17-14-9-5-4-8-12(13)14/h1-10H
    Synonyms: 2-Phenyl-4H-chromen-4-on | NSC19028 | 2-phenyl-4H-chromone | AKOS000603572 | HMS2269O06 | EN300-18246169 | NCGC000909...
  3. Riluzole, Sodium channel alpha subunit blocker
    Cas Number: 1744-22-5        Compound CID:  5070
    Formula:  C8H5F3N2OS        Molecular Weight: 234.2
    IUPAC Name:  6-(trifluoromethoxy)-1,3-benzothiazol-2-amine
    SMILES:  C1=CC2=C(C=C1OC(F)(F)F)SC(=N2)N
    InChIKey: FTALBRSUTCGOEG-UHFFFAOYSA-N
    InChI:  InChI=1S/C8H5F3N2OS/c9-8(10,11)14-4-1-2-5-6(3-4)15-7(12)13-5/h1-3H,(H2,12,13)
    Synonyms: 6-(trifluoromethoxy)-1,3-benzothiazol-2-amine | 6-(trifluoromethoxy)benzo[d]thiazol-2-amine | Bio1_001394 | RILUZOLE ...
  4. 1-[2-(Trifluoromethyl)phenyl]imidazole, Channel blocker of TRPV2
    Cas Number: 25371-96-4        Compound CID:  1359
    Formula:  C10H7F3N2        Molecular Weight: 212.18
    IUPAC Name:  1-[2-(trifluoromethyl)phenyl]imidazole
    SMILES:  C1=CC=C(C(=C1)C(F)(F)F)N2C=CN=C2
    InChIKey: WZBWBNCQUTXYEL-UHFFFAOYSA-N
    InChI:  InChI=1S/C10H7F3N2/c11-10(12,13)8-3-1-2-4-9(8)15-6-5-14-7-15/h1-7H
    Synonyms: NCGC00016047-03 | 1-(2-trifluoromethylphenyl) imidazole | 1-(2-Trifluoromethylphenyl)imidazole | 2-(trifluoromethyl)p...
  5. 4-Aminopyridine, Voltage-gated potassium channel blocker
      Grade & Purity: 
    • ≥98%
    Cas Number: 504-24-5        EC Number: 207-987-9
    Formula:  C5H6N2        Molecular Weight: 94.11
    IUPAC Name:  pyridin-4-amine
    SMILES:  C1=CN=CC=C1N
    InChIKey: NUKYPUAOHBNCPY-UHFFFAOYSA-N
    InChI:  InChI=1S/C5H6N2/c6-5-1-3-7-4-2-5/h1-4H,(H2,6,7)
    Synonyms: AI3-52547 | Amaya | Avitrol | Dalfampridine (USAN) | Fampridine-PR | BH3B64OKL9 | DTXCID003870 | p-amino pyridine | B...
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