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hGPR91 antagonist 1 - 10mM in DMSO, high purity , CAS No.1314796-00-3(DMSO)

COA

Grade & Purity:

10mM in DMSO

Cas Number: 1314796-00-3(DMSO)
Molecular Weight: 529.53

In stock

Item Number

H655892

Grouped product items
SKU	Size	Availability	Price	Qty
H655892-1ml	1ml	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$286.90

View related series

Compound libraries (12325) GPCR/G Protein (3172) Succinate Receptor 1 (5)

Basic Description

Specifications & Purity	10mM in DMSO
Biochemical and Physiological Mechanisms	HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC 50 of 7 μM.
Storage Temp	Store at -80°C
Shipped In	Ice chest + Ice pads This product requires cold chain shipping. Ground and other economy services are not available.
Product Description	HGPR91 antagonist 1 is a potent and selective small molecule hGPR91 antagonist with an IC 50 of 7 μM In Vivo HGPR91 antagonist 1 leads to 59, 76% inhibition of ΔMAP at 2, 4 hours and has shown rat plasma protein binding 99%. HGPR91 antagonist 1 has engaged the target under the in vivo condition. HGPR91 antagonist 1 has clearance (CL) of 0.2 nmol/min/mg of RLM . MCE has not independently confirmed the accuracy of these methods. They are for reference only. Animal Model: Wistar rats Dosage: 100 mg/kg Administration: I.p.; 2 and 4 hours Result: Led to 59 and 76% inhibition of ΔMAP at 2 and 4 hours. IC50& Target:IC50: 7 μM (HGPR91)

Associated Targets(Human)

SUCNR1 Tchem Succinate receptor 1 (1 Activities)

Discover Target: SUCNR1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

Smiles	CC(C1=CC=C(C=C1)C2=CC(=C(C=C2)F)C(F)(F)F)NC(=O)CC3=CC=C(C=C3)C4=NC5=C(C=CC=N5)C=C4
Molecular Weight	529.53

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

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