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DSTBULET, Agonist of δ receptor, CAS No.111035-56-4, Agonist of δ receptor

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rp173911
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rp173911-500μg
500μg
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$1,334.90
rp173911-1mg
1mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,334.90
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δ receptor Agonist (40)

Basic Description

Product Name DSTBULET, Agonist of δ receptor, CAS No.111035-56-4
Synonyms (Ser(2)(O-t-butyl)-leu(5))enkephalyl-thr(6) | Leu(5) enkephalin, ser(2)(O-tert-butyl)-thr(6) | Tyr-D-Ser(O-t-Bu)-Gly-Phe-Leu-Thr | Tyr-D-Ser(OtBu)-Gly-Phe-Leu-Thr | Q27077122 | Dstbulet | DTXSID40149447 | BDBM50019053 | Tyr-ser(O-tert-Bu)-gly-phe-leu-thr
Grade Moligand™
Specifications & Purity Moligand™
Action Type AGONIST
Mechanism of action Agonist of δ receptor

Taxonomic Classification

Taxonomy Tree

Kingdom Organic compounds
Superclass Organic acids and derivatives
Class Carboxylic acids and derivatives
Subclass Amino acids, peptides, and analogues
Intermediate Tree Nodes Peptides
Direct Parent Oligopeptides
Alternative Parents Tyrosine and derivatives  Phenylalanine and derivatives  Leucine and derivatives  N-acyl-L-alpha-amino acids  Alpha amino acid amides  Amphetamines and derivatives  1-hydroxy-2-unsubstituted benzenoids  Aralkylamines  Beta hydroxy acids and derivatives  N-acyl amines  Amino acids  Secondary carboxylic acid amides  Secondary alcohols  Dialkyl ethers  Carboxylic acids  Monocarboxylic acids and derivatives  Monoalkylamines  Organopnictogen compounds  Hydrocarbon derivatives  Carbonyl compounds  Organic oxides  
Molecular Framework Aromatic homomonocyclic compounds
Substituents Alpha-oligopeptide - Tyrosine or derivatives - Phenylalanine or derivatives - Leucine or derivatives - N-acyl-alpha-amino acid - N-acyl-alpha amino acid or derivatives - N-acyl-l-alpha-amino acid - Alpha-amino acid amide - Alpha-amino acid or derivatives - Amphetamine or derivatives - N-substituted-alpha-amino acid - 1-hydroxy-2-unsubstituted benzenoid - Aralkylamine - Beta-hydroxy acid - Phenol - Monocyclic benzene moiety - Fatty acyl - Benzenoid - Fatty amide - Hydroxy acid - N-acyl-amine - Amino acid or derivatives - Amino acid - Secondary carboxylic acid amide - Carboxamide group - Secondary alcohol - Monocarboxylic acid or derivatives - Carboxylic acid - Ether - Dialkyl ether - Organonitrogen compound - Amine - Organic nitrogen compound - Carbonyl group - Organic oxygen compound - Hydrocarbon derivative - Organic oxide - Organopnictogen compound - Primary aliphatic amine - Primary amine - Organooxygen compound - Alcohol - Aromatic homomonocyclic compound
Description This compound belongs to the class of organic compounds known as oligopeptides. These are organic compounds containing a sequence of between three and ten alpha-amino acids joined by peptide bonds.
External Descriptors Not available

Associated Targets(Human)

OPRD1 Tclin Delta-type opioid receptor (0 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
OPRM1 Tclin Mu opioid receptor (19785 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID
OPRD1 Tclin Delta opioid receptor (15096 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID

Associated Targets(non-human)

Cavia porcellus (23802 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID
Mus musculus (284745 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID

Mechanisms of Action

Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References

Storage and Shipping

CAS 111035-56-4

Certificates(CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Genetic information

Alternate Names (Ser(2)(O-t-butyl)-leu(5))enkephalyl-thr(6) | Leu(5) enkephalin, ser(2)(O-tert-butyl)-thr(6) | Tyr-D-Ser(O-t-Bu)-Gly-Phe-Leu-Thr | Tyr-D-Ser(OtBu)-Gly-Phe-Leu-Thr | Q27077122 | Dstbulet | DTXSID40149447 | BDBM50019053 | Tyr-ser(O-tert-Bu)-gly-phe-leu-thr
Reference
  • 1. Kinetics and inhibition of recombinant human cystathionine gamma-lyase. Toward the rational control of transsulfuration., The Journal of biological chemistry, Steegborn, C C and 7 more authors.
  • 2. Generation and initial analysis of more than 15,000 full-length human and mouse cDNA sequences., Proceedings of the National Academy of Sciences of the United States of America, Strausberg, Robert L RL and 83 more authors.
  • 3. Genomic basis of cystathioninuria (MIM 219500) revealed by multiple mutations in cystathionine gamma-lyase (CTH)., Human genetics, Wang, Jian J and Hegele, Robert A RA.
  • 4. Cloning and nucleotide sequence of human liver cDNA encoding for cystathionine gamma-lyase., Biochemical and biophysical research communications, Lu, Y Y, O'Dowd, B F BF, Orrego, H H and Israel, Y Y.
  • 5. Single nucleotide polymorphism in CTH associated with variation in plasma homocysteine concentration., Clinical genetics, Wang, J J, Huff, A M AM, Spence, J D JD and Hegele, R A RA.
  • 6. Cystathionine gamma-lyase overexpression inhibits cell proliferation via a H2S-dependent modulation of ERK1/2 phosphorylation and p21Cip/WAK-1., The Journal of biological chemistry, Yang, Guangdong G, Cao, Kun K, Wu, Lingyun L and Wang, Rui R.
  • 7. The status, quality, and expansion of the NIH full-length cDNA project: the Mammalian Gene Collection (MGC)., Genome research, Gerhard, Daniela S DS and 115 more authors.
  • 8. Towards a proteome-scale map of the human protein-protein interaction network., Nature, Rual, Jean-François JF and 37 more authors.
  • 9. The DNA sequence and biological annotation of human chromosome 1., Nature, Gregory, S G SG and 178 more authors.
  • 10. Polymorphisms in one-carbon metabolism and trans-sulfuration pathway genes and susceptibility to bladder cancer., International journal of cancer, Moore, Lee E LE and 14 more authors. more

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