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Deltasonamide 1 TFA , CAS No.2235358-73-1

COA

Cas Number: 2235358-73-1
Molecular Weight: 761.27

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Item Number

D651265

Grouped product items
SKU	Size	Availability	Price
D651265-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$260.90
D651265-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$780.90
D651265-10mg	10mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,250.90

View related series

Metabolic Enzyme/Protease (4860) Nucleic Acid Metabolism (395) Phosphodiesterase (PDE) (252)

Basic Description

Biochemical and Physiological Mechanisms	Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a K D of 203 pM. Deltasonamide 1 can be used for the research of tumors.
Storage Temp	Store at 2-8°C,Desiccated
Shipped In	Wet ice This product requires cold chain shipping. Ground and other economy services are not available.
Product Description	Deltasonamide 1 TFA is a PDE6δ-KRas inhibitor. Deltasonamide 1 can inhibit PDE6δ-KRas with a K D of 203 pM. Deltasonamide 1 can be used for the research of tumors In Vitro Deltasonamide 1 can inhibit PDE6δ-KRas with a K D of 203 pM. Deltasonamide 1 binds to PDE6δ with up to 7 hydrogen bonds, resulting in picomolar affinity. Deltasonamide 1 strongly reduces proliferation. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Cell Proliferation AssayCell Line: RTCA of hPDAC cell lines Concentration: 0.375, 0.75, 1.5, 3, 6, 12 μM Incubation Time: 60 h Result: Inhibited proliferation of human pancreatic cancer cell lines. Form:Solid IC50& Target:KD: 203 pM (PDE6δ-KRas)

Names and Identifiers

Smiles	O=S(C1=CC=C(S(=O)(N(CC2=NC(NC)=NC=C2)CC3CCNCC3)=O)C=C1)(N(CC4=CC=C(Cl)C=C4)C5CCCC5)=O.O=C(O)C(F)(F)F
Molecular Weight	761.27

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