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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
BAY-899 |
36; BAY-899 | IC50 | > | 16 | uM | ALA4323794 | nM | Homo sapiens | |||
| 2. |
ALA4537998 |
33; BAY-298 | IC50 | > | 16 | uM | ALA4323794 | nM | Homo sapiens | |||
| 3. |
ALA4449797 |
1b | IC50 | > | 16500 | nM | ALA4323794 | nM | Homo sapiens | |||
| 4. |
ALA4471621 |
1a | IC50 | > | 16500 | nM | ALA4323794 | nM | Homo sapiens | |||
| 5. |
ALA4593222 |
1 | IC50 | > | 16500 | nM | ALA4323794 | nM | Homo sapiens | |||
| 6. |
BAY-899 |
36; BAY-899 | IC50 | > | 16 | uM | ALA5214241 | nM | Homo sapiens | |||
| 7. |
ALA4592872 |
EUB0000340 | IC50 | > | 16 | uM | ALA5214359 | nM | Homo sapiens | |||
| 8. |
ALA5281228 |
rac-1; ORG 274179-0 | IC50 | = | 17 | nM | ALA5256363 | 7.77 | nM | Homo sapiens | ||
| 9. |
ALA5275472 |
66 | Efficacy | = | 87 | % | ALA5256334 | % | Homo sapiens | |||
| 10. |
ALA5268829 |
69 | Efficacy | = | 83 | % | ALA5256334 | % | Homo sapiens | |||
| 11. |
ALA5286556 |
68 | Efficacy | = | 84 | % | ALA5256334 | % | Homo sapiens | |||
| 12. |
ALA5273361 |
8b | Efficacy | = | 88 | % | ALA5256334 | % | Homo sapiens |