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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA1253609 |
17 | IC50 | = | 3.83 | ug ml-1 | ALA4310817 | ug.mL-1 | Rattus norvegicus | |||
| 2. |
Shogaol |
8 | Activity | = | 111.6 | % | ALA4321773 | % | Rattus norvegicus | |||
| 3. |
(-)-Securinin |
securinine | Activity | = | 101.8 | % | ALA4321773 | % | Rattus norvegicus | |||
| 4. |
ALA4436897 |
5 | Activity | = | 101.1 | % | ALA4321773 | % | Rattus norvegicus | |||
| 5. |
ALA4452328 |
3 | Activity | = | 101.4 | % | ALA4321773 | % | Rattus norvegicus | |||
| 6. |
Shogaol |
8 | Activity | = | 138.7 | % | ALA4321772 | % | Rattus norvegicus | |||
| 7. |
(-)-Securinin |
securinine | Activity | = | 141.1 | % | ALA4321772 | % | Rattus norvegicus | |||
| 8. |
ALA4436897 |
5 | Activity | = | 172.7 | % | ALA4321772 | % | Rattus norvegicus | |||
| 9. |
ALA4452328 |
3 | Activity | = | 145.3 | % | ALA4321772 | % | Rattus norvegicus | |||
| 10. |
ALA4541923 |
24c; TG11-224 | CC50 | 0 | ALA4325407 | Not Determined | Rattus norvegicus | |||||
| 11. |
ALA4587876 |
24b; TG11-242 | CC50 | > | 50 | uM | ALA4325407 | nM | Rattus norvegicus | |||
| 12. |
ALA4537092 |
24a; TG11-228 | CC50 | > | 50 | uM | ALA4325407 | nM | Rattus norvegicus |