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# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. |
ALA4474064 |
65 | IC50 | = | 10.9 | uM | ALA4310796 | 4.96 | nM | Trypanosoma brucei brucei | ||
2. |
ALA4589788 |
64 | IC50 | = | 2.83 | uM | ALA4310794 | 5.55 | nM | Trypanosoma brucei brucei | ||
3. |
ALA4550259 |
63 | IC50 | = | 8.48 | uM | ALA4310794 | 5.07 | nM | Trypanosoma brucei brucei | ||
4. |
ALA1720939 |
SID56373877 | IC50 | = | 0.937 | uM | ALA4310784 | 6.03 | nM | Trypanosoma brucei brucei | ||
5. |
2-Phenylbenzo[d]isothiazol-3(2H)-one |
7 | IC50 | = | 0.092 | uM | ALA4310784 | 7.04 | nM | Trypanosoma brucei brucei | ||
6. |
ALA4436808 |
20g | pEC50 | = | 7.7 | ALA4325174 | 7.70 | nM | Trypanosoma brucei brucei | |||
7. |
ALA4514007 |
20r | EC50 | = | 152 | nM | ALA4325174 | 6.82 | nM | Trypanosoma brucei brucei | ||
8. |
ALA4436808 |
20g | Activity | 0 | ALA4325203 | Not Active | Trypanosoma brucei brucei | |||||
9. |
ALA4436808 |
20g | Activity | 0 | ALA4325202 | Active | Trypanosoma brucei brucei | |||||
10. |
ALA4514007 |
20r | pEC99 | < | 6 | ALA4325197 | Trypanosoma brucei brucei | |||||
11. |
ALA4436808 |
20g | pEC99 | >= | 6 | ALA4325197 | Trypanosoma brucei brucei | |||||
12. |
ALA4514007 |
20r | pEC50 | < | 6 | ALA4325196 | nM | Trypanosoma brucei brucei |