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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
CHDI 00390576 |
22 | INH | < | 25 | % | ALA4311074 | % | Homo sapiens | |||
| 2. |
ALA4437833 |
16 | INH | < | 25 | % | ALA4311074 | % | Homo sapiens | |||
| 3. |
Belzutifan |
2; PT2977 | Activity | 0 | ALA4312721 | Not Active | Homo sapiens | |||||
| 4. |
ALA304335 |
19l | Ki | = | 3 | nM | ALA4186984 | 8.52 | nM | Homo sapiens | ||
| 5. |
ALA303380 |
19k | Ki | = | 2 | nM | ALA4186984 | 8.70 | nM | Homo sapiens | ||
| 6. |
ALA304272 |
19j | Ki | = | 3 | nM | ALA4186984 | 8.52 | nM | Homo sapiens | ||
| 7. |
ALA293228 |
18f | Ki | = | 2 | nM | ALA4186984 | 8.70 | nM | Homo sapiens | ||
| 8. |
ALA3793277 |
29k | IC50 | = | 9.5 | nM | ALA4221048 | 8.02 | nM | Homo sapiens | ||
| 9. |
ALA4228089 |
(S)-42c | IC50 | = | 350 | nM | ALA4221048 | 6.46 | nM | Homo sapiens | ||
| 10. |
ALA4225709 |
(R)-42c | IC50 | = | 58 | nM | ALA4221048 | 7.24 | nM | Homo sapiens | ||
| 11. |
ALA4224781 |
42e | IC50 | = | 46 | nM | ALA4221048 | 7.34 | nM | Homo sapiens | ||
| 12. |
ALA4227282 |
42d | IC50 | = | 100 | nM | ALA4221048 | 7.00 | nM | Homo sapiens |