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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4283703 |
(+/-)-1 | Activity | 0 | ALA4256543 | Not Active | Rattus norvegicus | |||||
| 2. |
ALA1086654 |
4 | Imax | = | 1.02 | % | ALA4256538 | % | Rattus norvegicus | |||
| 3. |
ALA4290888 |
(2aR,4aS,9aS)-1 | Imax | = | 1.1 | % | ALA4256538 | % | Rattus norvegicus | |||
| 4. |
ALA4283703 |
(+/-)-1 | Imax | = | 1.08 | % | ALA4256538 | % | Rattus norvegicus | |||
| 5. |
Acetylcholine |
table I | EC50 | = | 110 | uM | ALA4256537 | nM | Rattus norvegicus | |||
| 6. |
ALA1086654 |
4 | EC50 | = | 21 | uM | ALA4256537 | 4.68 | nM | Rattus norvegicus | ||
| 7. |
ALA4290888 |
(2aR,4aS,9aS)-1 | EC50 | = | 4 | uM | ALA4256537 | 5.40 | nM | Rattus norvegicus | ||
| 8. |
ALA4283703 |
(+/-)-1 | EC50 | = | 9.9 | uM | ALA4256537 | 5.00 | nM | Rattus norvegicus | ||
| 9. |
(±)-Epibatidine |
9 | Ki | 0 | ALA4154650 | Not Determined | Rattus norvegicus | |||||
| 10. |
ALA4176790 |
14o | Ki | = | 101 | 10'3nM | ALA4154650 | nM | Rattus norvegicus | |||
| 11. |
ALA4165509 |
14n | Ki | 0 | ALA4154650 | Not Determined | Rattus norvegicus | |||||
| 12. |
ALA4173434 |
14m | Ki | = | 5.1 | 10'3nM | ALA4154650 | 5.29 | nM | Rattus norvegicus |