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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
TDI-11861 |
33; TDI-11861 | IC50 | = | 5.5 | nM | ALA5218090 | 8.26 | nM | Rattus norvegicus | ||
| 2. |
ALA5220647 |
32 | IC50 | = | 10.8 | nM | ALA5218090 | 7.97 | nM | Rattus norvegicus | ||
| 3. |
ALA5219443 |
31 | IC50 | = | 22.9 | nM | ALA5218090 | 7.64 | nM | Rattus norvegicus | ||
| 4. |
ALA5219579 |
30 | IC50 | = | 34.8 | nM | ALA5218090 | 7.46 | nM | Rattus norvegicus | ||
| 5. |
ALA5220685 |
29 | IC50 | = | 2.5 | nM | ALA5218090 | 8.60 | nM | Rattus norvegicus | ||
| 6. |
ALA5218552 |
28 | IC50 | = | 19.6 | nM | ALA5218090 | 7.71 | nM | Rattus norvegicus | ||
| 7. |
ALA5218702 |
27 | IC50 | = | 16.7 | nM | ALA5218090 | 7.78 | nM | Rattus norvegicus | ||
| 8. |
ALA5218615 |
26 | IC50 | = | 14.6 | nM | ALA5218090 | 7.84 | nM | Rattus norvegicus | ||
| 9. |
ALA5218878 |
25 | IC50 | = | 5.5 | nM | ALA5218090 | 8.26 | nM | Rattus norvegicus | ||
| 10. |
ALA5220632 |
24 | IC50 | = | 37.7 | nM | ALA5218090 | 7.42 | nM | Rattus norvegicus | ||
| 11. |
ALA5218698 |
23 | IC50 | = | 1.9 | nM | ALA5218090 | 8.72 | nM | Rattus norvegicus |