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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4752133 |
2 | CL | = | 0.175 | uL/min | ALA4672291 | uL/min | Rattus norvegicus | |||
| 2. |
ALA4788098 |
1 | CL | = | 0.334 | uL/min | ALA4672291 | uL/min | Rattus norvegicus | |||
| 3. |
ALA3780541 |
SYL930 | CL | = | 0.437 | uL/min | ALA4672291 | uL/min | Rattus norvegicus | |||
| 4. |
Fingolimod HCl |
FTY720 (1a) | CL | = | 0.95 | uL/min | ALA4672291 | uL/min | Rattus norvegicus | |||
| 5. |
ALA4752133 |
2 | Km | = | 23.6 | umol/L | ALA4672290 | nM | Rattus norvegicus | |||
| 6. |
ALA4788098 |
1 | Km | = | 48.37 | umol/L | ALA4672290 | nM | Rattus norvegicus | |||
| 7. |
ALA3780541 |
SYL930 | Km | = | 85.25 | umol/L | ALA4672290 | nM | Rattus norvegicus | |||
| 8. |
Fingolimod HCl |
FTY720 (1a) | Km | = | 64.6 | umol/L | ALA4672290 | nM | Rattus norvegicus | |||
| 9. |
ALA4752133 |
2 | Vmax | = | 4.13 | pmol/min | ALA4672289 | pmol/min | Rattus norvegicus | |||
| 10. |
ALA4788098 |
1 | Vmax | = | 16.15 | pmol/min | ALA4672289 | pmol/min | Rattus norvegicus | |||
| 11. |
ALA3780541 |
SYL930 | Vmax | = | 37.24 | pmol/min | ALA4672289 | pmol/min | Rattus norvegicus | |||
| 12. |
Fingolimod HCl |
FTY720 (1a) | Vmax | = | 61.3 | pmol/min | ALA4672289 | pmol/min | Rattus norvegicus |