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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4529955 |
19 | IC50 | = | 102.5 | nM | ALA4424133 | 6.99 | nM | Homo sapiens | ||
| 2. |
ALA4519811 |
18d | IC50 | = | 213.9 | nM | ALA4424133 | 6.67 | nM | Homo sapiens | ||
| 3. |
ALA4516515 |
18c | IC50 | = | 9.6 | nM | ALA4424133 | 8.02 | nM | Homo sapiens | ||
| 4. |
ALA4581972 |
18b | IC50 | = | 3 | nM | ALA4424133 | 8.52 | nM | Homo sapiens | ||
| 5. |
ALA4524568 |
15c | IC50 | < | 0.3 | nM | ALA4424133 | nM | Homo sapiens | |||
| 6. |
ALA4578043 |
16 | IC50 | > | 200 | nM | ALA4424133 | nM | Homo sapiens | |||
| 7. |
ALA4576727 |
15a | IC50 | = | 4.3 | nM | ALA4424133 | 8.37 | nM | Homo sapiens | ||
| 8. |
Gilteritinib |
GILTERITINIB | IC50 | = | 8.5 | nM | ALA4424133 | 8.07 | nM | Homo sapiens | ||
| 9. |
ALA4475960 |
13b | IC50 | > | 200 | nM | ALA4424133 | nM | Homo sapiens | |||
| 10. |
ALA4592943 |
13a | IC50 | > | 200 | nM | ALA4424133 | nM | Homo sapiens | |||
| 11. |
ALA4462288 |
11 | IC50 | > | 1000 | nM | ALA4424133 | nM | Homo sapiens |