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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4528598 |
1; ARD-61 | DC50 | = | 1 | nM | ALA4324997 | nM | Homo sapiens | |||
| 2. |
ALA4528598 |
1; ARD-61 | DC50 | = | 7.2 | nM | ALA4324996 | nM | Homo sapiens | |||
| 3. |
ALA4528598 |
1; ARD-61 | Activity | > | 90 | % | ALA4324995 | % | Homo sapiens | |||
| 4. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325023 | Homo sapiens | |||||
| 5. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325022 | Homo sapiens | |||||
| 6. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325021 | Homo sapiens | |||||
| 7. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325020 | Homo sapiens | |||||
| 8. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325019 | Homo sapiens | |||||
| 9. |
ARD-266 |
11; ARD-266 | Activity | 0 | ALA4325015 | Not Active | Homo sapiens | |||||
| 10. |
ARD-266 |
11; ARD-266 | FC | >= | 10 | ALA4325018 | Homo sapiens | |||||
| 11. |
ARD-266 |
11; ARD-266 | Activity | 0 | ALA4324998 | Dose-dependent effect | Homo sapiens | |||||
| 12. |
ARD-266 |
11; ARD-266 | Activity | 0 | ALA4324997 | Dose-dependent effect | Homo sapiens |