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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4533018 |
IM-93 | Activity | = | 91 | % | ALA4308013 | % | Homo sapiens | |||
| 2. |
ALA4576489 |
8b | Kd | = | 85 | nM | ALA4322871 | 7.07 | nM | Homo sapiens | ||
| 3. |
ALA4465866 |
8a | Kd | = | 109 | nM | ALA4322871 | 6.96 | nM | Homo sapiens | ||
| 4. |
ROCK inhibitor-2 |
16 | IC50 | = | 1 | nM | ALA4328711 | 9.00 | nM | Homo sapiens | ||
| 5. |
Staurosporine |
1 (Staurosporine) | IC50 | = | 2.84 | 10'-9M | ALA4328575 | 8.55 | nM | Homo sapiens | ||
| 6. |
Staurosporine |
1 (Staurosporine) | IC50 | = | 1.23 | 10'-9M | ALA4328574 | 8.91 | nM | Homo sapiens | ||
| 7. |
Staurosporine |
1 (Staurosporine) | Activity | < | 65 | % | ALA4328211 | % | Homo sapiens | |||
| 8. |
Staurosporine |
1 (Staurosporine) | Activity | < | 65 | % | ALA4328210 | % | Homo sapiens | |||
| 9. |
ALA4446405 |
7b; ASR352 | Activity | = | 101.79 | % | ALA4327847 | % | Homo sapiens | |||
| 10. |
ALA4438024 |
7a; NSC30049; NSC49L | Activity | = | 101.9 | % | ALA4327847 | % | Homo sapiens | |||
| 11. |
ALA4446405 |
7b; ASR352 | Activity | = | 105.25 | % | ALA4327846 | % | Homo sapiens | |||
| 12. |
ALA4438024 |
7a; NSC30049; NSC49L | Activity | = | 95.01 | % | ALA4327846 | % | Homo sapiens |