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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4583803 |
Ar5Y_4 | Kd | = | 1.38 | uM | ALA4330218 | 5.86 | nM | Homo sapiens | ||
| 2. |
ALA4544177 |
Ar5Y_3 | Kd | = | 3.13 | uM | ALA4330218 | 5.50 | nM | Homo sapiens | ||
| 3. |
ALA4458745 |
Ar5Y_2 | Kd | = | 3.14 | uM | ALA4330218 | 5.50 | nM | Homo sapiens | ||
| 4. |
ALA4436009 |
Ar5Y_1 | Kd | = | 3.39 | uM | ALA4330218 | 5.47 | nM | Homo sapiens | ||
| 5. |
ALA4205401 |
Fig 11, Cpd 1 | IC50 | < | 50 | nM | ALA4184946 | nM | Homo sapiens | |||
| 6. |
ALA4216328 |
Fig 11, Cpd 2 | IC50 | < | 50 | nM | ALA4184946 | nM | Homo sapiens | |||
| 7. |
ALA5201066 |
39 | Activity | 0 | ALA5155940 | NA | Homo sapiens | |||||
| 8. |
ALA5092744 |
L7 | Kd | = | 3.34 | nM | ALA5225070 | 8.48 | nM | Homo sapiens | ||
| 9. |
ALA4461906 |
3 | Activity | 0 | ALA4307480 | Not Active | Homo sapiens | |||||
| 10. |
ALA4532684 |
2 | Activity | 0 | ALA4307480 | Not Active | Homo sapiens | |||||
| 11. |
ALA4438020 |
1 | Activity | 0 | ALA4307480 | Not Active | Homo sapiens | |||||
| 12. |
ALA4793446 |
66 | Kd | = | 1.66 | mM | ALA4670080 | nM | Homo sapiens |