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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
6-Bromocoumarin-3-carboxylic Acid |
15, UBP608 | IC50 | = | 68 | uM | ALA4309027 | 4.17 | nM | Homo sapiens | ||
| 2. |
ALA5181502 |
45e | INH | = | 12.04 | % | ALA5132338 | % | Homo sapiens | |||
| 3. |
ALA5181502 |
45e | INH | = | 16.16 | % | ALA5132338 | % | Homo sapiens | |||
| 4. |
ALA5181502 |
45e | INH | = | 14.95 | % | ALA5132338 | % | Homo sapiens | |||
| 5. |
ALA305187 |
(+/-)-ifenprodil | INH | = | 28.84 | % | ALA5132338 | % | Homo sapiens | |||
| 6. |
SAGE-718 |
DALZANEMDOR | Emax | = | 86 | % | ALA5136767 | % | Homo sapiens | |||
| 7. |
SAGE-718 |
DALZANEMDOR | EC50 | = | 150 | nM | ALA5136765 | 6.82 | nM | Homo sapiens | ||
| 8. |
ALA5092058 |
EUB0001556 | %max | = | 200 | % | ALA5145421 | % | Homo sapiens | |||
| 9. |
ALA5092058 |
EUB0001556 | EC50 | > | 30 | uM | ALA5145396 | nM | Homo sapiens | |||
| 10. |
ALA4460335 |
3 | IC50 | > | 10 | uM | ALA4339651 | nM | Homo sapiens | |||
| 11. |
ALA4475155 |
4 | IC50 | > | 10 | uM | ALA4339651 | nM | Homo sapiens | |||
| 12. |
ALA2426097 |
26 | INH | = | 21 | % | ALA2427687 | % | Homo sapiens |