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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
2-((1-(2-Fluoro-4-((4-(1-isopropyl-1H-pyrazol-4-yl)-5-methylpyrimidin-2-yl)amino)phenyl)piperidin-4-yl)(methyl)amino)ethan-1-ol |
18e | IC50 | = | 578.4 | nM | ALA4323959 | 6.24 | nM | Homo sapiens | ||
| 2. |
2-((1-(2-Fluoro-4-((4-(1-isopropyl-1H-pyrazol-4-yl)-5-methylpyrimidin-2-yl)amino)phenyl)piperidin-4-yl)(methyl)amino)ethan-1-ol |
18e | IC50 | = | 112.3 | nM | ALA4323947 | 6.95 | nM | Homo sapiens | ||
| 3. |
ALA5269603 |
5 | IC50 | = | 169 | nM | ALA5252499 | 6.77 | nM | Homo sapiens | ||
| 4. |
ALA5268459 |
4 | IC50 | = | 218 | nM | ALA5252499 | 6.66 | nM | Homo sapiens | ||
| 5. |
ALA5271559 |
3 | IC50 | > | 10000 | nM | ALA5252499 | nM | Homo sapiens | |||
| 6. |
ALA5279787 |
2 | IC50 | = | 116 | nM | ALA5252499 | 6.94 | nM | Homo sapiens | ||
| 7. |
ALA5270549 |
CEE321; 1 | IC50 | = | 54 | nM | ALA5252499 | 7.27 | nM | Homo sapiens | ||
| 8. |
ALA5269603 |
5 | IC50 | = | 2169 | nM | ALA5252493 | 5.66 | nM | Homo sapiens | ||
| 9. |
ALA5268459 |
4 | IC50 | = | 525 | nM | ALA5252493 | 6.28 | nM | Homo sapiens | ||
| 10. |
ALA5271559 |
3 | IC50 | > | 30000 | nM | ALA5252493 | nM | Homo sapiens | |||
| 11. |
ALA5279787 |
2 | IC50 | > | 30000 | nM | ALA5252493 | nM | Homo sapiens | |||
| 12. |
ALA5270549 |
CEE321; 1 | IC50 | = | 2349 | nM | ALA5252493 | 5.63 | nM | Homo sapiens |