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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA5271646 |
60 | IC50 | = | 50 | uM | ALA5263508 | 4.30 | nM | Homo sapiens | ||
| 2. |
ALA1964644 |
SID103905106 | Activity | 0 | ALA4482770 | Active | Homo sapiens | |||||
| 3. |
ALA4534968 |
DB2-114; DB4 | IC50 | = | 1.5 | uM | ALA4482760 | 5.82 | nM | Homo sapiens | ||
| 4. |
ALA4592322 |
DB2-082; DB2 | IC50 | = | 3 | uM | ALA4482760 | 5.52 | nM | Homo sapiens | ||
| 5. |
ALA4560825 |
DB2-113; DB3 | IC50 | = | 4.5 | uM | ALA4482760 | 5.35 | nM | Homo sapiens | ||
| 6. |
ALA1964644 |
SID103905106 | IC50 | = | 10 | uM | ALA4482760 | 5.00 | nM | Homo sapiens | ||
| 7. |
ALA4575072 |
DB2-001 | IC50 | = | 20 | uM | ALA4482760 | 4.70 | nM | Homo sapiens | ||
| 8. |
Fingolimod |
3 | IC50 | = | 6.3 | uM | ALA2444689 | 5.20 | nM | Homo sapiens | ||
| 9. |
ALA2441555 |
5 | IC50 | = | 10.4 | uM | ALA2444689 | 4.98 | nM | Homo sapiens | ||
| 10. |
ALA2441554 |
6 | IC50 | = | 3.8 | uM | ALA2444689 | 5.42 | nM | Homo sapiens | ||
| 11. |
ALA2441553 |
7 | IC50 | = | 9.7 | uM | ALA2444689 | 5.01 | nM | Homo sapiens | ||
| 12. |
ALA2441552 |
8 | IC50 | = | 13.8 | uM | ALA2444689 | 4.86 | nM | Homo sapiens |