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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA2430437 |
RGH 237 | Ratio Ki | > | 1800 | ALA2434790 | Rattus norvegicus | |||||
| 2. |
ALA20734 |
55 | Kd | = | 0.095 | nM | ALA3057572 | 10.02 | nM | Rattus norvegicus | ||
| 3. |
ALA20734 |
55 | Kd | = | 0.01 | nM | ALA3057571 | 11.00 | nM | Rattus norvegicus | ||
| 4. |
ALA42 |
clozapine | Ki | = | 134 | nM | ALA3057566 | 6.87 | nM | Rattus norvegicus | ||
| 5. |
ALA715 |
Olanzapine | Ki | = | 90 | nM | ALA3057566 | 7.05 | nM | Rattus norvegicus | ||
| 6. |
Haloperidol |
Haloperidol | Ki | = | 2.39 | nM | ALA3057566 | 8.62 | nM | Rattus norvegicus | ||
| 7. |
Domperidone |
Domperidone | Ki | = | 3.08 | nM | ALA3057566 | 8.51 | nM | Rattus norvegicus | ||
| 8. |
S33084 |
4x | Ki | = | 53.8 | nM | ALA3057566 | 7.27 | nM | Rattus norvegicus | ||
| 9. |
4-(2-Aminoethyl)benzene-1,2-diol |
Dopamine | IC50 | = | 582 | nM | ALA3057566 | 6.24 | nM | Rattus norvegicus | ||
| 10. |
quinpirole |
Quinpirole | IC50 | = | 454 | nM | ALA3057566 | 6.34 | nM | Rattus norvegicus | ||
| 11. |
ALA531 |
pergolide | IC50 | = | 5.59 | nM | ALA3057566 | 8.25 | nM | Rattus norvegicus | ||
| 12. |
(R)-(-)-Apomorphine |
apomorphine | IC50 | = | 69.5 | nM | ALA3057566 | 7.16 | nM | Rattus norvegicus |