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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4454100 |
16 | INH | = | 5.5 | % | ALA4309142 | % | Homo sapiens | |||
| 2. |
ALA4447975 |
(+/-)-4j | INH | <= | 50 | % | ALA4308650 | % | Homo sapiens | |||
| 3. |
ALA4447975 |
(+/-)-4j | pKi | < | 5 | ALA4308606 | nM | Homo sapiens | ||||
| 4. |
ALA4457754 |
(+/-)-4c | INH | <= | 50 | % | ALA4308650 | % | Homo sapiens | |||
| 5. |
ALA4572167 |
(+/-)-3c | INH | <= | 50 | % | ALA4308650 | % | Homo sapiens | |||
| 6. |
ALA4572167 |
(+/-)-3c | pKi | < | 5 | ALA4308606 | nM | Homo sapiens | ||||
| 7. |
ALA4528651 |
(+/-)-3b | INH | <= | 50 | % | ALA4308650 | % | Homo sapiens | |||
| 8. |
ALA4528651 |
(+/-)-3b | pKi | < | 5 | ALA4308606 | nM | Homo sapiens | ||||
| 9. |
ALA4472703 |
(+/-)-3a | INH | <= | 50 | % | ALA4308650 | % | Homo sapiens | |||
| 10. |
ALA4472703 |
(+/-)-3a | pKi | < | 5 | ALA4308606 | nM | Homo sapiens | ||||
| 11. |
ALA4457754 |
(+/-)-4c | pKi | < | 5 | ALA4308606 | nM | Homo sapiens | ||||
| 12. |
ALA4238634 |
11 | INH | < | 30 | % | ALA4232487 | % | Homo sapiens |