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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA5306577 |
EUB0002354 | Inhibition | = | -1.5 | % | ALA5304397 | % | Homo sapiens | |||
| 2. |
Ibudilast |
Ibudilast | IC50 | <= | 10 | uM | ALA5227532 | nM | Homo sapiens | |||
| 3. |
Anagrelide |
BL-4162A | IC50 | = | 0.9 | nM | ALA5256545 | 9.05 | nM | Homo sapiens | ||
| 4. |
ALA5283704 |
18; BCH24426 | IC50 | = | 32 | nM | ALA5256543 | 7.50 | nM | Homo sapiens | ||
| 5. |
Anagrelide |
BL-4162A | IC50 | = | 30 | nM | ALA5256543 | 7.52 | nM | Homo sapiens | ||
| 6. |
Lixazinone |
1 (lixazinone) | IC50 | = | 10 | nM | ALA5256543 | 8.00 | nM | Homo sapiens | ||
| 7. |
Cilostazol |
Cilostazol | IC50 | = | 200 | nM | ALA5256543 | 6.70 | nM | Homo sapiens | ||
| 8. |
Cilostamide |
Cilostamide, OPC-3689 | IC50 | = | 27 | nM | ALA5256543 | 7.57 | nM | Homo sapiens | ||
| 9. |
Vesnarinone |
9 | IC50 | = | 6200 | nM | ALA5256543 | 5.21 | nM | Homo sapiens | ||
| 10. |
ALA66522 |
36 | IC50 | = | 70 | nM | ALA5256543 | 7.16 | nM | Homo sapiens | ||
| 11. |
Quazinone (Ro 13-6438) |
4 | IC50 | = | 580 | nM | ALA5256543 | 6.24 | nM | Homo sapiens | ||
| 12. |
Zardaverine |
zardaverine | IC50 | = | 580 | nM | ALA5256543 | 6.24 | nM | Homo sapiens |