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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4442651 |
5 | Activity | 0 | ALA4323783 | Dose-dependent effect | Homo sapiens | |||||
| 2. |
ALA4442651 |
5 | Activity | 0 | ALA4323775 | Not Active | Homo sapiens | |||||
| 3. |
ALA4593469 |
10 | IC50 | > | 1000 | nM | ALA4323771 | nM | Homo sapiens | |||
| 4. |
ALA4469125 |
8 | IC50 | > | 1000 | nM | ALA4323771 | nM | Homo sapiens | |||
| 5. |
ALA4454796 |
7 | IC50 | > | 1000 | nM | ALA4323771 | nM | Homo sapiens | |||
| 6. |
ALA4575577 |
6 | IC50 | > | 1000 | nM | ALA4323771 | nM | Homo sapiens | |||
| 7. |
ALA4442651 |
5 | IC50 | = | 18.9 | nM | ALA4323771 | 7.72 | nM | Homo sapiens | ||
| 8. |
ALA4534088 |
4 | IC50 | > | 1000 | nM | ALA4323771 | nM | Homo sapiens | |||
| 9. |
ALA4446073 |
1 | IC50 | = | 294 | nM | ALA4323771 | 6.53 | nM | Homo sapiens | ||
| 10. |
ALA4461668 |
Cpd D | IC50 | = | 1.39 | nM | ALA4323772 | 8.86 | nM | Homo sapiens | ||
| 11. |
ALA3289606 |
3 | Activity | > | 5000 | nM | ALA4323770 | nM | Homo sapiens | |||
| 12. |
ALA4582414 |
Cpd E | Activity | > | 5000 | nM | ALA4323770 | nM | Homo sapiens |