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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA3786952 |
101 | IC50 | = | 0.16 | uM | ALA4223302 | 6.80 | nM | Homo sapiens | ||
| 2. |
2,3-Pyridinedicarboxylic acid |
QUIN | IC50 | > | 10000 | uM | ALA5229135 | nM | Homo sapiens | |||
| 3. |
2,6-Pyridinedicarboxylic acid |
47 | IC50 | = | 250 | uM | ALA5229135 | nM | Homo sapiens | |||
| 4. |
2,5-Pyridinedicarboxylic acid |
2 | IC50 | = | 1900 | uM | ALA5229135 | nM | Homo sapiens | |||
| 5. |
2,4-Pyridinedicarboxylic acid(PCA) |
32 | IC50 | = | 4.7 | uM | ALA5229135 | 5.33 | nM | Homo sapiens | ||
| 6. |
JIB-04 |
SID524082 | IC50 | = | 0.34 | uM | ALA5237466 | 6.47 | nM | Homo sapiens | ||
| 7. |
ALA5277662 |
7 | IC50 | = | 2.3 | uM | ALA5237417 | 5.64 | nM | Homo sapiens | ||
| 8. |
2,4-Pyridinedicarboxylic acid(PCA) |
32 | IC50 | = | 3 | uM | ALA5237417 | 5.52 | nM | Homo sapiens | ||
| 9. |
ALA2169917 |
55 | IC50 | = | 0.11 | uM | ALA5231386 | 6.96 | nM | Homo sapiens | ||
| 10. |
ALA3108956 |
8 | IC50 | = | 6.4 | uM | ALA5231386 | 5.19 | nM | Homo sapiens | ||
| 11. |
8-Hydroxyquinoline-5-carboxylic Acid |
SID85736331 | IC50 | = | 0.2 | uM | ALA5216092 | 6.70 | nM | Homo sapiens | ||
| 12. |
ALA1933775 |
15 | IC50 | = | 0.9 | uM | ALA5141172 | 6.05 | nM | Homo sapiens |