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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
KJ Pyr 9 |
5a | Activity | = | 100 | % | ALA4234733 | % | Homo sapiens | |||
| 2. |
KJ Pyr 9 |
5a | Kd | = | 6.5 | nM | ALA4234737 | 8.19 | nM | Homo sapiens | ||
| 3. |
KJ Pyr 9 |
5a | IC50 | = | 1 | uM | ALA4234738 | 6.00 | nM | Homo sapiens | ||
| 4. |
ALA4240401 |
5b | Activity | = | 106 | % | ALA4234733 | % | Homo sapiens | |||
| 5. |
ALA4240401 |
5b | IC50 | = | 3 | uM | ALA4234738 | 5.52 | nM | Homo sapiens | ||
| 6. |
ALA4247460 |
5c | Activity | = | 79 | % | ALA4234733 | % | Homo sapiens | |||
| 7. |
ALA4247460 |
5c | IC50 | = | 30 | uM | ALA4234738 | 4.52 | nM | Homo sapiens | ||
| 8. |
ALA4241092 |
5d | Activity | = | 0 | % | ALA4234733 | % | Homo sapiens | |||
| 9. |
ALA4241092 |
5d | IC50 | > | 100 | uM | ALA4234738 | nM | Homo sapiens | |||
| 10. |
ALA4245253 |
5e | Activity | = | 41 | % | ALA4234733 | % | Homo sapiens | |||
| 11. |
ALA4245253 |
5e | IC50 | = | 40 | uM | ALA4234738 | 4.40 | nM | Homo sapiens | ||
| 12. |
ALA4244986 |
5f | Activity | = | 55 | % | ALA4234733 | % | Homo sapiens |