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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4247506 |
2a | INH | = | 0 | % | ALA4230180 | % | Homo sapiens | |||
| 2. |
ALA3736320 |
15 | INH | = | 29 | % | ALA4230180 | % | Homo sapiens | |||
| 3. |
ALA3125821 |
17 | Activity | 0 | ALA4233966 | Active | Homo sapiens | |||||
| 4. |
ALA4207014 |
19 | INH | = | 13 | % | ALA4191105 | % | Homo sapiens | |||
| 5. |
ALA4209540 |
4b | Activity | = | 112 | % | ALA4178089 | % | Homo sapiens | |||
| 6. |
ALA2171133 |
22 | IC50 | < | 15 | nM | ALA5252711 | nM | Homo sapiens | |||
| 7. |
ALA2171134 |
23 | IC50 | < | 15 | nM | ALA5252711 | nM | Homo sapiens | |||
| 8. |
GSK2593074A |
21 | IC50 | < | 15 | nM | ALA5252711 | nM | Homo sapiens | |||
| 9. |
ALA2171128 |
2 | IC50 | < | 15 | nM | ALA5252711 | nM | Homo sapiens | |||
| 10. |
ALA2171131 |
20 | IC50 | < | 15 | nM | ALA5252711 | nM | Homo sapiens | |||
| 11. |
ALA2171145 |
34 | IC50 | = | 17 | nM | ALA5252711 | 7.77 | nM | Homo sapiens | ||
| 12. |
ALA4441909 |
22b | Activity | 0 | ALA4425434 | Active | Homo sapiens |