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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4277021 |
4k | Activity | > | 80 | % | ALA4270731 | % | Homo sapiens | |||
| 2. |
ALA4533018 |
IM-93 | Activity | = | 78 | % | ALA4308069 | % | Homo sapiens | |||
| 3. |
ALA4576489 |
8b | Kd | = | 60 | nM | ALA4322794 | 7.22 | nM | Homo sapiens | ||
| 4. |
ALA4465866 |
8a | Kd | = | 44 | nM | ALA4322794 | 7.36 | nM | Homo sapiens | ||
| 5. |
Staurosporine |
1 (Staurosporine) | IC50 | = | 6.62 | 10'-8M | ALA4328624 | 7.18 | nM | Homo sapiens | ||
| 6. |
Staurosporine |
1 (Staurosporine) | Activity | < | 65 | % | ALA4328260 | % | Homo sapiens | |||
| 7. |
ALA4446405 |
7b; ASR352 | Activity | = | 99.98 | % | ALA4327896 | % | Homo sapiens | |||
| 8. |
ALA4438024 |
7a; NSC30049; NSC49L | Activity | = | 100.52 | % | ALA4327896 | % | Homo sapiens | |||
| 9. |
ALA4251324 |
30 | IC50 | > | 10000 | nM | ALA4233414 | nM | Homo sapiens | |||
| 10. |
ALA4245507 |
28 | IC50 | > | 10000 | nM | ALA4233414 | nM | Homo sapiens | |||
| 11. |
PDGFRα kinase inhibitor 1 |
15i | Activity | = | 92 | % | ALA4230971 | % | Homo sapiens | |||
| 12. |
ALA4247506 |
2a | INH | = | 5 | % | ALA4230235 | % | Homo sapiens |