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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
UNC2025 |
11, UNC2025 | IC50 | = | 4.38 | nM | ALA4276357 | 8.36 | nM | Homo sapiens | ||
| 2. |
UNC4203 |
19 | IC50 | = | 8.4 | nM | ALA4276357 | 8.08 | nM | Homo sapiens | ||
| 3. |
ALA1098827 |
Trp-Ox | Kd | = | 13 | uM | ALA4326996 | 4.89 | nM | Homo sapiens | ||
| 4. |
ALA4460719 |
3 | IC50 | = | 4.1 | uM | ALA4309193 | 5.39 | nM | Homo sapiens | ||
| 5. |
ALA1896117 |
SID74373667 | IC50 | > | 50 | uM | ALA4309193 | nM | Homo sapiens | |||
| 6. |
ALA4533018 |
IM-93 | Activity | = | 100 | % | ALA4308088 | % | Homo sapiens | |||
| 7. |
Belizatinib (TSR-011) |
36 | IC50 | < | 0.003 | uM | ALA4330193 | nM | Homo sapiens | |||
| 8. |
Altiratinib |
ALTIRATINIB | IC50 | = | 0.008 | uM | ALA4330193 | 8.08 | nM | Homo sapiens | ||
| 9. |
TrkA-IN-1 |
39 | IC50 | = | 25 | uM | ALA4330193 | 4.60 | nM | Homo sapiens | ||
| 10. |
ALA4469569 |
40 | IC50 | > | 81 | uM | ALA4330193 | nM | Homo sapiens | |||
| 11. |
ALA4584074 |
45 | IC50 | = | 7.1 | uM | ALA4330193 | 5.15 | nM | Homo sapiens | ||
| 12. |
ALA4443139 |
46 | IC50 | = | 2.3 | uM | ALA4330193 | 5.64 | nM | Homo sapiens |