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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
BI 78D3 |
12, BI-78D3 | Ki | = | 2.3 | 10^-6M | ALA5152482 | 5.64 | nM | Rattus norvegicus | ||
| 2. |
ALA2151190 |
1 | INH | = | 50 | % | ALA2155183 | % | Rattus norvegicus | |||
| 3. |
ALA2151190 |
1 | IC50 | = | 1 | uM | ALA2155182 | 6.00 | nM | Rattus norvegicus | ||
| 4. |
ALA2000337 |
SID493510 | INH | = | 45 | % | ALA2155151 | % | Rattus norvegicus | |||
| 5. |
ALA2151193 |
4 | INH | = | 47 | % | ALA2155151 | % | Rattus norvegicus | |||
| 6. |
ALA2151192 |
3 | INH | = | 100 | % | ALA2155151 | % | Rattus norvegicus | |||
| 7. |
ALA2151191 |
2(-), (-)-zuonin A | INH | = | 50 | % | ALA2155151 | % | Rattus norvegicus | |||
| 8. |
ALA2151286 |
11 | IC50 | 0 | ALA2155150 | Not Active | Rattus norvegicus | |||||
| 9. |
ALA2151285 |
10 | IC50 | 0 | ALA2155150 | Not Active | Rattus norvegicus | |||||
| 10. |
Furaltadone |
SID482725 | IC50 | 0 | ALA2155150 | Not Active | Rattus norvegicus | |||||
| 11. |
ALA2000337 |
SID493510 | IC50 | = | 57 | uM | ALA2155150 | 4.24 | nM | Rattus norvegicus | ||
| 12. |
ALA1492532 |
SID26664743 | IC50 | 0 | ALA2155150 | Not Active | Rattus norvegicus |