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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4531700 |
MC-FCQR-QK | Ki | > | 10000 | nM | ALA4330019 | nM | Homo sapiens | |||
| 2. |
ALA4530379 |
MCoTI-II | Ki | > | 10000 | nM | ALA4330019 | nM | Homo sapiens | |||
| 3. |
ALA4564063 |
MC-FCQR | Ki | > | 10000 | nM | ALA4330019 | nM | Homo sapiens | |||
| 4. |
DKFZ‐251 |
11; DKFZ-251 | Activity | 0 | ALA4201858 | Not Active | Homo sapiens | |||||
| 5. |
DKFZ‐251 |
11; DKFZ-251 | IC50 | = | 73 | uM | ALA4201844 | 4.14 | nM | Homo sapiens | ||
| 6. |
ALA4206734 |
39 | IC50 | > | 0.5 | uM | ALA4201844 | nM | Homo sapiens | |||
| 7. |
ALA4227614 |
36b | IC50 | = | 4.1 | uM | ALA4222616 | 5.39 | nM | Homo sapiens | ||
| 8. |
ALA4228178 |
36a | IC50 | = | 0.11 | uM | ALA4222616 | 6.96 | nM | Homo sapiens | ||
| 9. |
ALA4227339 |
35b | IC50 | = | 7 | uM | ALA4222616 | 5.16 | nM | Homo sapiens | ||
| 10. |
ALA4228441 |
35a | IC50 | = | 0.048 | uM | ALA4222616 | 7.32 | nM | Homo sapiens | ||
| 11. |
ALA4227602 |
34b | IC50 | = | 2.8 | uM | ALA4222616 | 5.55 | nM | Homo sapiens | ||
| 12. |
ALA4227658 |
34a | IC50 | = | 0.45 | uM | ALA4222616 | 6.35 | nM | Homo sapiens |