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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA1098827 |
Trp-Ox | Kd | = | 3.8 | uM | ALA4326995 | 5.42 | nM | Homo sapiens | ||
| 2. |
Indolo[2,1-b]quinazoline-6,12-dione |
1 (Tryptanthrine) | Kd | = | 7.2 | uM | ALA4326995 | 5.14 | nM | Homo sapiens | ||
| 3. |
ALA4460719 |
3 | IC50 | = | 14 | uM | ALA4309192 | 4.85 | nM | Homo sapiens | ||
| 4. |
ALA1896117 |
SID74373667 | IC50 | > | 50 | uM | ALA4309192 | nM | Homo sapiens | |||
| 5. |
ALA4573890 |
G755-0360 | IC50 | = | 358.6 | nM | ALA4308450 | 6.45 | nM | Homo sapiens | ||
| 6. |
ALA4467890 |
G755-0459 | IC50 | = | 20000 | nM | ALA4308450 | 4.70 | nM | Homo sapiens | ||
| 7. |
ALA4466913 |
G755-0551 | IC50 | = | 20000 | nM | ALA4308450 | 4.70 | nM | Homo sapiens | ||
| 8. |
ALA4466570 |
G755-0331 | IC50 | = | 10000 | nM | ALA4308450 | 5.00 | nM | Homo sapiens | ||
| 9. |
ALA4450466 |
G755-0467 | IC50 | = | 10000 | nM | ALA4308450 | 5.00 | nM | Homo sapiens | ||
| 10. |
ALA4468419 |
2a; L365-0764 | IC50 | = | 423.2 | nM | ALA4308450 | 6.37 | nM | Homo sapiens | ||
| 11. |
ALA4536149 |
L365-0799 | IC50 | = | 778 | nM | ALA4308450 | 6.11 | nM | Homo sapiens | ||
| 12. |
ALA4448594 |
L365-1408 | IC50 | = | 20000 | nM | ALA4308450 | 4.70 | nM | Homo sapiens |