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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA5271233 |
18 | INH | 0 | ALA5225785 | Active | % | Homo sapiens | ||||
| 2. |
ALA5271233 |
18 | INH | 0 | ALA5225784 | Active | % | Homo sapiens | ||||
| 3. |
ALA5289039 |
23; 4EGI-1 | Kd | = | 25 | uM | ALA5232213 | 4.60 | nM | Homo sapiens | ||
| 4. |
ALA5180948 |
102 | pIC50 | = | 7.5 | ALA5137679 | 7.50 | nM | Homo sapiens | |||
| 5. |
ALA5183975 |
101 | pIC50 | = | 8.5 | ALA5137679 | 8.50 | nM | Homo sapiens | |||
| 6. |
ALA5181488 |
100 | pIC50 | = | 8.1 | ALA5137679 | 8.10 | nM | Homo sapiens | |||
| 7. |
ALA5203720 |
99 | pIC50 | = | 8.1 | ALA5137679 | 8.10 | nM | Homo sapiens | |||
| 8. |
ALA5171562 |
98 | pIC50 | = | 7.5 | ALA5137679 | 7.50 | nM | Homo sapiens | |||
| 9. |
ALA5206647 |
97 | pIC50 | = | 7.8 | ALA5137679 | 7.80 | nM | Homo sapiens | |||
| 10. |
ALA5197975 |
96 | pIC50 | = | 7.1 | ALA5137679 | 7.10 | nM | Homo sapiens | |||
| 11. |
ALA5205835 |
95 | pIC50 | = | 7.4 | ALA5137679 | 7.40 | nM | Homo sapiens | |||
| 12. |
ALA5195407 |
94 | pIC50 | = | 7.6 | ALA5137679 | 7.60 | nM | Homo sapiens |