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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4248427 |
154 | IC50 | = | 43 | nM | ALA4229775 | 7.37 | nM | Homo sapiens | ||
| 2. |
Captopril |
Captopril | IC50 | = | 6.3 | nM | ALA4229775 | 8.20 | nM | Homo sapiens | ||
| 3. |
Omapatrilat |
1a, BMS-186716 | Ki | = | 0.016 | nM | ALA4269910 | 10.80 | nM | Homo sapiens | ||
| 4. |
Omapatrilat |
1a, BMS-186716 | Ki | = | 0.015 | nM | ALA4269909 | 10.82 | nM | Homo sapiens | ||
| 5. |
ALA4294217 |
Omapatrilat Dimer | IC50 | = | 1.8 | uM | ALA4269908 | 5.75 | nM | Homo sapiens | ||
| 6. |
ALA4294217 |
Omapatrilat Dimer | IC50 | = | 2.1 | uM | ALA4269907 | 5.68 | nM | Homo sapiens | ||
| 7. |
ALA4294217 |
Omapatrilat Dimer | IC50 | = | 2.8 | uM | ALA4269906 | 5.55 | nM | Homo sapiens | ||
| 8. |
Omapatrilat |
1a, BMS-186716 | IC50 | = | 1 | nM | ALA4269906 | 9.00 | nM | Homo sapiens | ||
| 9. |
ALA4294217 |
Omapatrilat Dimer | IC50 | = | 2.2 | uM | ALA4269905 | 5.66 | nM | Homo sapiens | ||
| 10. |
Omapatrilat |
1a, BMS-186716 | IC50 | = | 2 | nM | ALA4269905 | 8.70 | nM | Homo sapiens | ||
| 11. |
ALA4202767 |
56 | Activity | <= | 25 | % | ALA4187164 | % | Homo sapiens | |||
| 12. |
Microginin 527 |
4 | IC50 | = | 31 | uM | ALA4144750 | 4.51 | nM | Homo sapiens |