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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4516396 |
10a | IC50 | > | 1000 | nM | ALA4327427 | nM | Homo sapiens | |||
| 2. |
ALA131 |
Prednisolone | IC50 | > | 1000 | nM | ALA4327427 | nM | Homo sapiens | |||
| 3. |
ALA4467278 |
9d | IC50 | > | 1000 | nM | ALA4327427 | nM | Homo sapiens | |||
| 4. |
ALA4449031 |
9b | IC50 | = | 780 | nM | ALA4327427 | 6.11 | nM | Homo sapiens | ||
| 5. |
ALA113332 |
9g | INH | 0 | ALA4275695 | Not Active | % | Homo sapiens | ||||
| 6. |
ALA4278637 |
VPC-3033 | INH | 0 | ALA4275695 | Not Active | % | Homo sapiens | ||||
| 7. |
CHDI 00390576 |
22 | INH | < | 25 | % | ALA4311093 | % | Homo sapiens | |||
| 8. |
ALA4437833 |
16 | INH | < | 25 | % | ALA4311093 | % | Homo sapiens | |||
| 9. |
ALA4513808 |
14, Single Atropisomer | IC50 | > | 10 | uM | ALA4324497 | nM | Homo sapiens | |||
| 10. |
ALA4175305 |
9 | Activity | 0 | ALA4137965 | Not Active | Homo sapiens | |||||
| 11. |
ALA4175305 |
9 | INH | 0 | ALA4137994 | Not Active | % | Homo sapiens | ||||
| 12. |
ALA4175305 |
9 | Activity | 0 | ALA4137984 | Not Active | Homo sapiens |