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| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
ALA4290371 |
25a; SOMCL-286 | IC50 | > | 1000 | nM | ALA4271721 | nM | Homo sapiens | |||
| 2. |
Poziotinib (HM781-36B) |
POZIOTINIB | IC50 | = | 5.3 | nM | ALA4271185 | 8.28 | nM | Homo sapiens | ||
| 3. |
Canertinib (CI-1033) |
18 | IC50 | = | 30 | nM | ALA4271185 | 7.52 | nM | Homo sapiens | ||
| 4. |
ALA2347958 |
BIBW2992 | IC50 | = | 14 | nM | ALA4271185 | 7.85 | nM | Homo sapiens | ||
| 5. |
AV 412 |
SID137276039 | IC50 | = | 19 | nM | ALA4271185 | 7.72 | nM | Homo sapiens | ||
| 6. |
ALA2110732 |
5 | IC50 | = | 45.7 | nM | ALA4271185 | 7.34 | nM | Homo sapiens | ||
| 7. |
ALA4294264 |
4 | IC50 | = | 1.036 | uM | ALA4271177 | 5.99 | nM | Homo sapiens | ||
| 8. |
ALA4286374 |
3 | IC50 | = | 0.096 | uM | ALA4271177 | 7.02 | nM | Homo sapiens | ||
| 9. |
ALA4290869 |
2; A-10 | IC50 | = | 19 | nM | ALA4271177 | 7.72 | nM | Homo sapiens | ||
| 10. |
Lapatinib |
GW-572016 | IC50 | = | 9.2 | nM | ALA4271177 | 8.04 | nM | Homo sapiens | ||
| 11. |
MD2-TLR4-IN-1 |
22m | INH | 0 | ALA4304898 | Not Active | % | Homo sapiens | ||||
| 12. |
ALA4533018 |
IM-93 | Activity | = | 92 | % | ALA4307799 | % | Homo sapiens |