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CBP/p300-IN-10 - 98%, high purity , CAS No.2259641-71-7

COA

Grade & Purity:

≥98%

Cas Number: 2259641-71-7
Molecular Weight: 537.48

In stock

Item Number

C648970

Grouped product items
SKU	Size	Availability	Price	Qty
C648970-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$450.90
C648970-5mg	5mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$1,450.90

View related series

Epigenetics (1496) Histone Acetyltransferase (79) Histone Modification (1379)

Basic Description

Specifications & Purity	≥98%
Biochemical and Physiological Mechanisms	CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer.
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads This product requires cold chain shipping. Ground and other economy services are not available.
Product Description	CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer In Vitro CBP/p300-IN-10 (example 84) (0-1 μM; 3 h) inhibit H3K27Ac activity in LK2 cells with an IC 50 of 22 nM. CBP/p300-IN-10 (38 nM-10 mM; 3 days) has inhibitory activity against LK2 and TE-8. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Cell Proliferation AssayCell Line: LK2 and TE-8 Concentration: 38 nM-10 mM Incubation Time: 3 days Result: Inhibited LK2 and TE-8 with GI 50 s of 97.163 nM and 152.484 nM, respectively. Form:Solid IC50& Target:EP300 26 nM (IC 50 ) CREBBP 39 nM (IC 50 )

Names and Identifiers

Smiles	O=C(N1[C@H](C[C@H](C1)F)C(NC2=CC=C(NN=C3)C3=N2)=O)C4(C5=CC=C(C=C5)OC(F)F)CCC(F)(CC4)F
Molecular Weight	537.48

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):

Analytical Chart:

Chemical and Physical Properties

Solubility	DMSO : 10.5 mg/mL (19.54 mM; ultrasonic and warming and heat to 80°C)

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