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AZD3778 , CAS No.1032129-23-9, Antagonist of CCR3;Antagonist of H 1 receptor;Channel blocker of K v11.1

COA COA
In stock
Item Number
A607865
Grouped product items
SKU Size
Availability
 Price Qty
A607865-5mg
5mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$1,000.90
A607865-25mg
25mg
Available within 8-12 weeks(?)
Production requires sourcing of materials. We appreciate your patience and understanding.
$2,000.90
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View related series
CCR3 Antagonist (18) H1 receptor Antagonist (64) Kv11.1 Channel blocker (13)

Basic Description

Synonyms AZD-3778 [WHO-DD] | 4-[4-(3,4-dichlorophenoxy)piperidin-1-yl]-N-(4-methylphenyl)sulfonylpiperidine-1-carboxamide | AZD3778 | AZD-3778 | UNII-9BC2MUG4A8 | 9BC2MUG4A8 | BDBM50394155 | N-((4-(3,4-Dichlorophenoxy)(1,4'-bipiperidin)-1'-yl)carbonyl)-4-methylben
Specifications & Purity Moligand™
Grade Moligand™
Action Type ANTAGONIST, CHANNEL BLOCKER
Mechanism of action Antagonist of CCR3;Antagonist of H 1 receptor;Channel blocker of K v11.1

Associated Targets(Human)

CCR3 Tchem C-C chemokine receptor type 3 (5 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
HRH1 Tclin Histamine H1 receptor (4 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
KCNH2 Tclin Potassium voltage-gated channel subfamily H member 2 (1 Activities)
Activity Type Activity Value -log(M) Mechanism of Action Activity Reference Publications (PubMed IDs)
HRH1 Tclin Histamine H1 receptor (7573 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID
KCNH2 Tclin HERG (29587 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID
CCR3 Tchem C-C chemokine receptor type 3 (1666 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID

Associated Targets(non-human)

Canis familiaris (36305 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID
Rattus norvegicus (775804 Activities)
Activity Type Relation Activity value Units Action Type Journal PubMed Id doi Assay Aladdin ID

Mechanisms of Action

Mechanism of Action Action Type target ID Target Name Target Type Target Organism Binding Site Name References

Names and Identifiers

IUPAC Name 4-[4-(3,4-dichlorophenoxy)piperidin-1-yl]-N-(4-methylphenyl)sulfonylpiperidine-1-carboxamide
INCHI InChI=1S/C24H29Cl2N3O4S/c1-17-2-5-21(6-3-17)34(31,32)27-24(30)29-12-8-18(9-13-29)28-14-10-19(11-15-28)33-20-4-7-22(25)23(26)16-20/h2-7,16,18-19H,8-15H2,1H3,(H,27,30)
InChIKey QVLZVRFIGXNZMN-UHFFFAOYSA-N
Smiles Cc1ccc(cc1)S(=O)(=O)NC(=O)N1CCC(CC1)N1CCC(CC1)Oc1ccc(c(c1)Cl)Cl
Isomeric SMILES CC1=CC=C(C=C1)S(=O)(=O)NC(=O)N2CCC(CC2)N3CCC(CC3)OC4=CC(=C(C=C4)Cl)Cl
PubChem CID 11753159

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Solution Calculators

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