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AS2717638 - 10mM in DMSO, high purity , CAS No.2148339-28-8(DMSO), Antagonist of LPA 5 receptor

COA

Grade & Purity:

Moligand™

10mM in DMSO

Cas Number: 2148339-28-8(DMSO)
Molecular Weight: 447.48

In stock

Item Number

A655490

Grouped product items
SKU	Size	Availability	Price	Qty
A655490-1ml	1ml	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$429.90

View related series

Compound libraries (12325) GPCR/G Protein (3172) LPL Receptor (113)

Basic Description

Specifications & Purity	Moligand™, 10mM in DMSO
Biochemical and Physiological Mechanisms	AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC 50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE 2 -, PGF 2α -, and AMPA-induced allodynia.
Storage Temp	Store at -80°C
Shipped In	Ice chest + Ice pads This product requires cold chain shipping. Ground and other economy services are not available.
Grade	Moligand™
Action Type	ANTAGONIST
Mechanism of action	Antagonist of LPA 5 receptor
Product Description	AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC 50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE 2 -, PGF 2α -, and AMPA-induced allodynia IC50& Target:IC50: 38 nM (hLPA5)

Associated Targets(Human)

LPAR5 Tchem Lysophosphatidic acid receptor 5 (1 Activities)

Discover Target: LPAR5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Names and Identifiers

Smiles	CC1=CC2=C(C=C1)ON=C2N3C=C(C4=CC(=C(C=C4C3=O)OC)OC)C(=O)N5CCCCC5
Molecular Weight	447.48

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

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