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Anamorelin - ≥98%, high purity , CAS No.249921-19-5

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Anamorelin - ≥98%, high purity , CAS No.249921-19-5

COA

Grade & Purity:

≥98%

Cas Number: 249921-19-5
Molecular Weight: 546.7
PubChem CID: 9828911

In stock

Item Number

A125440

Grouped product items
SKU	Size	Availability	Price
A125440-1mg	1mg	Available within 8-12 weeks(?) Production requires sourcing of materials. We appreciate your patience and understanding.	$17.90
A125440-5mg	5mg	3	$68.90
A125440-10mg	10mg	3	$98.90
A125440-50mg	50mg	3	$224.90

View related series

Class A GPCR (4138) GHSR (22) GPCR/G Protein (3172)

Basic Description

Synonyms	RC-1291 \| CCG-269985 \| UNII-6MUC9717YK \| HY-14734 \| RC-1291;ONO-7643 \| ST-1291 \| UNII-DD5RBA1NKF \| Q20707542 \| RC-1291 \| AKOS030526752 \| BCP06108 \| 2-Methyl-4-(2-phenyldiazenyl)phenol \| Anamorelin \| ANAMORELIN [WHO-DD] \| DB06645 \| CCG-5137 \| RC 1291 \| DD5
Specifications & Purity	≥98%
Biochemical and Physiological Mechanisms	Anamorelin hydrochloride is the orally bioavailable hydrochloride salt of a synthetic, small-molecule ghrelin mimetic with appetite-stimulating and anabolic activities. Anamorelin binds to and stimulates the growth hormone secretagogue re
Storage Temp	Store at -20°C
Shipped In	Ice chest + Ice pads This product requires cold chain shipping. Ground and other economy services are not available.
Product Description	Anamorelin(RC1291; ONO-7643) is a synthetic orally active ghrelin receptor agonist which is under development for the management of non-small lung cancer associated cachexia/anorexia.

Taxonomic Classification

Taxonomy Tree

Kingdom Organic compounds
- Superclass Organic acids and derivatives
  - Class Carboxylic acids and derivatives
    - Subclass Amino acids, peptides, and analogues
      - Level5 Peptides
        Level6 Dipeptides

Kingdom	Organic compounds
Superclass	Organic acids and derivatives
Class	Carboxylic acids and derivatives
Subclass	Amino acids, peptides, and analogues
Intermediate Tree Nodes	Peptides
Direct Parent	Dipeptides
Alternative Parents	3-benzylpiperidines N-acyl-alpha amino acids and derivatives Tryptamines and derivatives Alpha amino acid amides 3-alkylindoles Piperidinecarboxamides N-acylpiperidines Substituted pyrroles Benzene and substituted derivatives Heteroaromatic compounds Tertiary carboxylic acid amides Carboxylic acid hydrazides Secondary carboxylic acid amides Azacyclic compounds Hydrocarbon derivatives Carbonyl compounds Monoalkylamines Organic oxides
Molecular Framework	Aromatic heteropolycyclic compounds
Substituents	Alpha-dipeptide - N-acyl-alpha amino acid or derivatives - 3-benzylpiperidine - Benzylpiperidine - Alpha-amino acid amide - Triptan - Alpha-amino acid or derivatives - 3-alkylindole - Indole - Indole or derivatives - N-acyl-piperidine - 3-piperidinecarboxamide - Piperidinecarboxamide - Substituted pyrrole - Benzenoid - Piperidine - Monocyclic benzene moiety - Tertiary carboxylic acid amide - Pyrrole - Heteroaromatic compound - Secondary carboxylic acid amide - Amino acid or derivatives - Carboxamide group - Carboxylic acid hydrazide - Organoheterocyclic compound - Azacycle - Primary amine - Organic oxygen compound - Organic nitrogen compound - Primary aliphatic amine - Organic oxide - Carbonyl group - Amine - Hydrocarbon derivative - Organonitrogen compound - Organooxygen compound - Aromatic heteropolycyclic compound
Description	This compound belongs to the class of organic compounds known as dipeptides. These are organic compounds containing a sequence of exactly two alpha-amino acids joined by a peptide bond.
External Descriptors	Not available
1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61. DOI: 10.1186/s13321-016-0174-y

Associated Targets(non-human)

Hdac6 Histone deacetylase 6 (222 Activities)

Discover Target: Hdac6

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

rep Replicase polyprotein 1ab (378 Activities)

Discover Target: rep

Activity Type	Relation	Activity value	Units	Action Type	Journal	PubMed Id	doi	Assay Aladdin ID

Mechanisms of Action

Mechanism of Action	Action Type	target ID	Target Name	Target Type	Target Organism	Binding Site Name	References

Names and Identifiers

IUPAC Name	2-amino-N-[(2R)-1-[(3R)-3-benzyl-3-[dimethylamino(methyl)carbamoyl]piperidin-1-yl]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methylpropanamide
INCHI	InChI=1S/C31H42N6O3/c1-30(2,32)28(39)34-26(18-23-20-33-25-15-10-9-14-24(23)25)27(38)37-17-11-16-31(21-37,29(40)36(5)35(3)4)19-22-12-7-6-8-13-22/h6-10,12-15,20,26,33H,11,16-19,21,32H2,1-5H3,(H,34,39)/t26-,31-/m1/s1
InChIKey	VQPFSIRUEPQQPP-MXBOTTGLSA-N
Smiles	CC(C)(C(=O)NC(CC1=CNC2=CC=CC=C21)C(=O)N3CCCC(C3)(CC4=CC=CC=C4)C(=O)N(C)N(C)C)N
Isomeric SMILES	CC(C)(C(=O)N[C@H](CC1=CNC2=CC=CC=C21)C(=O)N3CCC[C@](C3)(CC4=CC=CC=C4)C(=O)N(C)N(C)C)N
Molecular Weight	546.7
Reaxy-Rn	13610248
Reaxys-RN_link_address	https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=13610248&ln=

Certificates（CoA,COO,BSE/TSE and Analysis Chart)

C of A & Other Certificates(BSE/TSE, COO):

Analytical Chart:

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1 results found

Lot Number	Certificate Type	Date	Item
I1609064	Certificate of Analysis	May 06, 2022	A125440

Chemical and Physical Properties

Solubility	DMSO
Molecular Weight	546.700 g/mol
XLogP3	2.800
Hydrogen Bond Donor Count	3
Hydrogen Bond Acceptor Count	5
Rotatable Bond Count	9
Exact Mass	546.332 Da
Monoisotopic Mass	546.332 Da
Topological Polar Surface Area	115.000 Å²
Heavy Atom Count	40
Formal Charge	0
Complexity	904.000
Isotope Atom Count	0
Defined Atom Stereocenter Count	2
Undefined Atom Stereocenter Count	0
Defined Bond Stereocenter Count	0
Undefined Bond Stereocenter Count	0
The total count of all stereochemical bonds	0
Covalently-Bonded Unit Count	1

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